Target Details
| UniProt AC | Q92918 |
|---|---|
| Gene Symbol | MAP4K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 225
- Clinical molecules 20
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (225)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
KOZFSFOOLUUIGY
|
6.3 | Kd | 88 | Yes | |
ARIDQNLHGPTVRV
|
6.3 | IC50 | 2 | — | |
AWKURTHTBAHLFJ
|
6.3 | IC50 | 2 | — | |
AZBCOCFKWZMQEJ
|
6.3 | IC50 | 2 | — | |
BBDMTVSVTWJQRA
|
6.3 | IC50 | 2 | — | |
BOMAZLQSSNNLAL
|
6.3 | IC50 | 2 | — | |
BXCYQVYUVRSMEO
|
6.3 | IC50 | 2 | — | |
BXRRZXRRYWPPRB
|
6.3 | IC50 | 2 | — | |
CEPCFYXGKVUSIE
|
6.3 | IC50 | 2 | — | |
CZYMIYVLJPMDKR
|
6.3 | IC50 | 2 | — | |
DCXQWYPQOMBAAM
|
6.3 | IC50 | 2 | — | |
DNSFNVWZLXWEIP
|
6.3 | IC50 | 2 | — | |
DSLFYWXOXHQCHX
|
6.3 | IC50 | 2 | — | |
GCIYNSCGYKCNRO
|
6.3 | IC50 | 2 | — | |
GPLMABVCEUFRFE
|
6.3 | IC50 | 2 | — | |
HZINCYNTSLFHIX
|
6.3 | IC50 | 2 | — | |
IISORMHFXQMHMH
|
6.3 | IC50 | 2 | — | |
IKKAOLZAHXWOGL
|
6.3 | IC50 | 2 | — | |
IRSFVELJVAKOKE
|
6.3 | IC50 | 2 | — | |
JBYRKKLGKRYYEB
|
6.3 | IC50 | 2 | — | |
JMNAJBKCXDWWFM
|
6.3 | IC50 | 2 | — | |
JRFVVGICARMPKA
|
6.3 | IC50 | 2 | — | |
JTZWLDGXHLBJLE
|
6.3 | IC50 | 2 | — | |
KRORJRNMSXNFRV
|
6.3 | IC50 | 2 | — | |
LBBPWLTWVVPJDU
|
6.3 | IC50 | 2 | — | |
LIVKHBBLMAFTFP
|
6.3 | IC50 | 2 | — | |
MAPGSKUWLDLVLP
|
6.3 | IC50 | 2 | — | |
MEZFXRCCCIIGIW
|
6.3 | IC50 | 2 | — | |
MKOUWRINCHLWSP
|
6.3 | IC50 | 2 | — | |
MNOLIHFFGYKXGE
|
6.3 | IC50 | 2 | — | |
MWUGCRIZPOMKMV
|
6.3 | IC50 | 2 | — | |
NAEBTWZBUODUEA
|
6.3 | IC50 | 2 | — | |
NBXVVYPBTMZIFQ
|
6.3 | IC50 | 2 | — | |
NHUNQBFMIZILLQ
|
6.3 | IC50 | 2 | — | |
OJKGBJDSLMQYOV
|
6.3 | IC50 | 2 | — | |
OWMRLFMYSUGJHS
|
6.3 | IC50 | 2 | — | |
OXDNNQYYISTXOB
|
6.3 | IC50 | 2 | — | |
PCLWCWPEGAQJBO
|
6.3 | IC50 | 2 | — | |
PMOGQHUXHONLRB
|
6.3 | IC50 | 2 | — | |
POUWYQSQNNTBKE
|
6.3 | IC50 | 2 | — | |
PPLCHDXBJPYXNY
|
6.3 | IC50 | 2 | — | |
PXCMMEQZVRGOBR
|
6.3 | IC50 | 2 | — | |
QFADKPXVEQNUDC
|
6.3 | IC50 | 2 | — | |
QXMYTSARCQSHKZ
|
6.3 | IC50 | 2 | — | |
QZLYZRALGDJSAC
|
6.3 | IC50 | 2 | — | |
RUHSHSFQBWSFOU
|
6.3 | IC50 | 2 | — | |
SPVRYWSSDGGGFK
|
6.3 | IC50 | 2 | — | |
SRAMWKCEWIPKEV
|
6.3 | IC50 | 2 | — | |
STXHTXUTWCUJHH
|
6.3 | IC50 | 2 | — |