Target Details
| UniProt AC | Q92918 |
|---|---|
| Gene Symbol | MAP4K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 225
- Clinical molecules 20
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (225)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XZXHXSATPCNXJR
|
7.5 | Kd | 165 | Yes | |
NHLRQGPSAURBBL
|
7.4 | IC50 | 3 | — | |
ORQCQXMGDYAIOI
|
7.4 | Ki | 6 | — | |
DTHDBWPUQXSBEE
|
7.4 | IC50 | 3 | — | |
OQCCQWBVUGOVBA
|
7.4 | Ki | 2 | — | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
KTEIFNKAUNYNJU
|
7.4 | Kd | 114 | — | |
YAPIPGOLZSTISM
|
7.4 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.4 | Kd | 154 | — | |
PIQCTGMSNWUMAF
|
7.4 | Kd | 137 | Yes | |
SEJGTFPOEJWEGG
|
7.4 | Kd | 149 | — | |
ZNRKSAWCBMXCBN
|
7.3 | IC50 | 3 | — | |
LQUUWQNDKXYUCK
|
7.3 | IC50 | 2 | — | |
LRINILBKXCVIMV
|
7.3 | IC50 | 3 | — | |
QVLFEWNYZXVCHO
|
7.3 | IC50 | 3 | — | |
ZZNHNGWYLUNNCT
|
7.3 | IC50 | 3 | — | |
DSXXEELGXBCYNQ
|
7.3 | IC50 | 28 | Yes | |
XCAXLCSQKKQKHA
|
7.2 | IC50 | 3 | — | |
HZYIMGKDYXEJDM
|
7.2 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
GCIKSSRWRFVXBI
|
7.1 | Kd | 109 | Yes | |
ZUJPITIYCZFUQQ
|
7.1 | IC50 | 3 | — | |
IAYGCINLNONXHY
|
7.1 | Kd | 50 | — | |
WTTUTRXPNFTTPC
|
7.1 | IC50 | 3 | — | |
JNCFZEVZRYWROV
|
7.1 | IC50 | 3 | — | |
DJWRSWJVUXTDII
|
7.0 | IC50 | 2 | — | |
YXFNNHJWPFANTQ
|
7.0 | IC50 | 3 | — | |
JWNPDZNEKVCWMY
|
7.0 | Kd | 57 | Yes | |
FRGXLZSKZPLLON
|
7.0 | Ki | 2 | — | |
IWFMUUASEIUTAN
|
7.0 | Ki | 2 | — | |
FKWAGVCCEZPSSL
|
7.0 | Ki | 3 | — | |
SOQDSWCPJNRWBD
|
7.0 | IC50 | 2 | — | |
FTBMREIZHCLTPN
|
6.9 | IC50 | 3 | — | |
KDKUVYLMPJIGKA
|
6.9 | Kd | 91 | Yes | |
SXGLKAJWKHWEPI
|
6.9 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
OYONTEXKYJZFHA
|
6.8 | Kd | 69 | Yes | |
HWXVIOGONBBTBY
|
6.8 | Kd | 27 | — | |
CTQLDDHACGXLAE
|
6.7 | Ki | 2 | — | |
XKFTZKGMDDZMJI
|
6.7 | Kd | 64 | Yes | |
BLLJUCXNHUVEHL
|
6.7 | IC50 | 3 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
VAARYSWULJUGST
|
6.7 | Kd | 119 | Yes | |
LOLPPWBBNUVNQZ
|
6.7 | Kd | 97 | Yes | |
HENRITOGWFFGGA
|
6.6 | Ki | 2 | — | |
MWKSRKSEWLRPBL
|
6.6 | Kd | 1075 | — | |
WVUNYSQLFKLYNI
|
6.6 | Kd | 46 | Yes | |
VCZPJHYQIPIKSV
|
6.6 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
6.5 | Kd | 43 | — | |
VRQMAABPASPXMW
|
6.5 | Kd | 10 | — |