Target Details
| UniProt AC | Q92918 |
|---|---|
| Gene Symbol | MAP4K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 225
- Clinical molecules 20
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (225)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHLFOJOOBSNVFP
|
8.3 | Ki | 2 | — | |
HSEDUERTEYTVOT
|
8.2 | IC50 | 2 | — | |
NRNCXXANURQNKO
|
8.2 | IC50 | 2 | — | |
BSBZFPBEYMSVPJ
|
8.1 | IC50 | 2 | — | |
KGMSWMZCIQWBHX
|
8.1 | IC50 | 3 | — | |
GFEVOBQWEKTOLR
|
8.1 | Ki | 2 | — | |
FRBVUOIUPMIQTN
|
8.1 | IC50 | 2 | — | |
ROEUNIAWGRPMCW
|
8.1 | IC50 | 2 | — | |
WUSZGZSHIMXCHY
|
8.1 | IC50 | 2 | — | |
RVSSNRBUPQUIEG
|
8.0 | IC50 | 5 | — | |
JBGWDRMZKMTPOT
|
8.0 | IC50 | 3 | — | |
PSZVRCRTXCCMNS
|
8.0 | Ki | 3 | — | |
KCVUUZPGZKJPAG
|
8.0 | IC50 | 2 | — | |
NSSDJHYKLWNDFG
|
8.0 | IC50 | 2 | — | |
JWBXEWFBXJNXBU
|
7.9 | Ki | 4 | — | |
VCCYOHCOICDUFL
|
7.9 | IC50 | 2 | — | |
NGGXDEMZRGKNHG
|
7.9 | IC50 | 2 | — | |
NSSDJHYKLWNDFG
|
7.9 | IC50 | 2 | — | |
LURPXFLMWSMKCY
|
7.9 | IC50 | 2 | — | |
VQYASORGHMGXQV
|
7.9 | IC50 | 2 | — | |
DZIXRHJRLCGYPK
|
7.8 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
7.8 | Kd | 55 | — | |
CTNPALGJUAXMMC
|
7.8 | Kd | 151 | — | |
GIRPCUVQSUVBEK
|
7.8 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
7.8 | Kd | 130 | Yes | |
WINHZLLDWRZWRT
|
7.8 | Kd | 201 | Yes | |
LJQVZLFSJBQAQB
|
7.8 | Ki | 2 | — | |
PPGUULSJUXLSJS
|
7.8 | IC50 | 2 | — | |
HEZSSKBBLQBTMF
|
7.8 | Ki | 4 | — | |
NXSJMRCTGYTSTK
|
7.8 | Kd | 200 | — | |
RKDKQDMKPCNZBL
|
7.8 | Ki | 2 | — | |
YBPNMUVFLXIRNQ
|
7.7 | IC50 | 2 | — | |
GCHHHYMKNXQPDG
|
7.7 | Ki | 2 | — | |
WECCALUSSAUMLJ
|
7.7 | IC50 | 2 | — | |
DSSNAGYVGTYAGH
|
7.7 | IC50 | 10 | — | |
STGJTJNMUPPEMH
|
7.7 | IC50 | 2 | — | |
TZPUNPWJLMOANL
|
7.6 | Ki | 6 | — | |
OSVUGUHRKMMBSE
|
7.6 | Kd | 170 | — | |
MOYRDZMEZHFJDU
|
7.6 | IC50 | 2 | — | |
UCUVIFYGOBXXKX
|
7.6 | IC50 | 2 | — | |
UKFXFNQXCIZAEM
|
7.6 | Ki | 2 | — | |
AIFRAZQXNNPZBV
|
7.6 | IC50 | 2 | — | |
GUUQXMDBAHSFGF
|
7.6 | IC50 | 4 | — | |
SUBYPZBREZXPCW
|
7.6 | Ki | 3 | — | |
YPUUKVINJSRXQN
|
7.6 | IC50 | 2 | — | |
RMYZEICXBRZXFD
|
7.6 | IC50 | 2 | — | |
CYJPFBCHYRZAJL
|
7.5 | IC50 | 3 | — | |
HUAPVUVLSXALII
|
7.5 | IC50 | 3 | — | |
JAOVTLWLVWUCIR
|
7.5 | IC50 | 2 | — | |
JKHBVOCOHYSWTQ
|
7.5 | Ki | 3 | — |