Target Details
| UniProt AC | Q92918 |
|---|---|
| Gene Symbol | MAP4K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 225
- Clinical molecules 20
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (225)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QFBHPPKNOIWKKI
|
10.8 | Ki | 2 | — | |
MXQDOIPMFYATOE
|
10.7 | Ki | 2 | — | |
DLNPTMIJPLMAGO
|
10.7 | Ki | 2 | — | |
YFRBRDWEJOCVAP
|
10.7 | Ki | 2 | — | |
WYARWPXUKWKBPH
|
10.4 | Ki | 2 | — | |
PIPGGBLVUJYMED
|
10.2 | Ki | 3 | — | |
XFXLQWRLVKKTHD
|
10.1 | Ki | 2 | — | |
XVKPIWUWUZOHIR
|
9.8 | Ki | 3 | — | |
CXIGTMXVRAHGKF
|
9.7 | IC50 | 2 | — | |
APVWQLVROLDAPP
|
9.5 | IC50 | 2 | — | |
PBRKEKVJQVXNEQ
|
9.3 | Ki | 2 | — | |
BQRDIEUIHZRWEL
|
9.3 | IC50 | 2 | — | |
KQCSODUJRAFWMC
|
9.2 | IC50 | 2 | — | |
NIJYDRGSAYMLLQ
|
9.2 | IC50 | 2 | — | |
APVWQLVROLDAPP
|
9.2 | IC50 | 2 | — | |
HGNARJFKBILTIL
|
9.2 | IC50 | 2 | — | |
NDXRAKYQSXBMOI
|
9.1 | IC50 | 2 | — | |
KQCSODUJRAFWMC
|
9.1 | IC50 | 2 | — | |
RWTXXGPUNDKBLW
|
9.1 | IC50 | 4 | — | |
RAHBGWKEPAQNFF
|
9.0 | Kd | 26 | — | |
WZCQVSWKOIATOS
|
9.0 | Ki | 2 | — | |
HFTWWDARPWZARK
|
9.0 | Ki | 3 | — | |
OXIQDNRCSPETQV
|
8.8 | IC50 | 2 | — | |
SIVPOEPNFMZRLH
|
8.8 | IC50 | 2 | — | |
PTIWUIAAGUMGEC
|
8.8 | Ki | 2 | — | |
FNVXHCSJUCJAGY
|
8.8 | Ki | 2 | — | |
HGNARJFKBILTIL
|
8.7 | IC50 | 2 | — | |
OEOIPLGKLNBGHY
|
8.7 | IC50 | 2 | — | |
LZYWVOKHWFMDJU
|
8.7 | Ki | 3 | — | |
OXIQDNRCSPETQV
|
8.7 | IC50 | 2 | — | |
OHKSBENCBXMGAT
|
8.7 | Ki | 2 | — | |
RVFYCRCCTDEQQD
|
8.6 | IC50 | 4 | — | |
UUVGYKHBHXIMIM
|
8.6 | IC50 | 2 | — | |
HPLDWJVEVHEYKM
|
8.6 | Ki | 2 | — | |
AOJDKUXYLYKLKG
|
8.6 | IC50 | 2 | — | |
PZWKQEQSYRXWEJ
|
8.6 | Ki | 2 | — | |
XSIMOSPDULMWPL
|
8.6 | IC50 | 3 | — | |
SYMONOSPGXDMMP
|
8.5 | IC50 | 2 | — | |
FRGYOMQWHFXVEU
|
8.4 | IC50 | 3 | — | |
QAJMXNDGDLWDAN
|
8.4 | IC50 | 3 | — | |
YLGMPWWMPCGYBF
|
8.4 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.4 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
8.4 | Kd | 213 | — | |
NGGXDEMZRGKNHG
|
8.3 | IC50 | 2 | — | |
OJPUQYTXGKTLEG
|
8.3 | IC50 | 2 | — | |
UQBOLKBTUZZWBP
|
8.3 | IC50 | 2 | — | |
UZPJPJXENPGVRI
|
8.3 | IC50 | 3 | — | |
WGUVBZYIVFUKTF
|
8.3 | IC50 | 2 | — | |
YKDKRNUADNJEHQ
|
8.3 | IC50 | 2 | — | |
BRNMCVNQMQLRHM
|
8.3 | IC50 | 3 | — |