Target Details
UniProt ACQ92831
Gene SymbolKAT2B
Protein NameHistone acetyltransferase KAT2B
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00583 (Acetyltransf_1) PF00439 (Bromodomain) PF06466 (PCAF_N)
Summary
  • Multi-target molecules 55
  • Clinical molecules 0
  • Avg pChEMBL 8.57
Top Co-occurrence Targets
Active Molecules (55)
InChIKey pChEMBL Type Targets Clinical
MCIGDGJLNSNEHL 10.7 Ki 2
VMOQDLYJQCKIKJ 10.4 Ki 2
KGYUNIZKDLZNSH 10.2 Ki 2
QSOFLSGOAZCHJA 10.2 Ki 2
RVZBXBUXJSRYKX 10.2 Ki 2
BWPNXWMSUALEOG 10.0 Ki 2
FDEZYLHCNMEOEN 10.0 Ki 2
SCGIEXBRKPZTKA 9.9 Ki 2
ZKFBZQMNSFITPE 9.8 Ki 2
TXWCNRCKXCEBOM 9.8 Ki 2
LRIDTLDQIOAIHB 9.7 Ki 2
OZNYMBYLDCQTSZ 9.7 Ki 2
CPXKHLLAEZFPHJ 9.7 Ki 2
NOVLKEPNLVCXTE 9.5 Ki 2
NVXRVMGLQIHNFH 9.5 Ki 2
UAIPDRJDVCRVGJ 9.5 Ki 2
RJLFPNSUABSXRV 9.4 Ki 2
TVOCBMWTXJRBLB 9.3 Ki 2
HINFIECYCWFNQN 9.3 Ki 2
SZITZWMQTGOBEC 9.3 Ki 2
YCXRPPJLAIUKFC 9.3 Ki 2
ZMOIEFSZHIKKFS 9.2 Ki 2
NLMIRYVVKHZQBM 9.2 Ki 2
GJZNKOBWUOEFNR 9.1 Ki 2
ZUUCCRLXECDZOE 9.1 Ki 2
GXUCAUXOCJIOPD 9.0 Ki 2
QOYJJEHJQBVOBM 9.0 Ki 2
CBPJBUBMKKGJMH 8.9 Ki 2
DAPYQEDLEDRHDE 8.6 Ki 2
DBBDEGULRIBGMX 8.6 Ki 2
AXPLCJNXRWLGIP 8.6 Ki 2
ZWGAQZOUQSOIQA 8.2 Ki 2
SLWLRRQDEFXBSW 8.2 Ki 2
UOQAFGWMKNIVAR 7.9 Kd 6
PYCNZAAZGQDRJG 7.9 IC50 2
CIUXKWFQVPTMEQ 7.8 Kd 3
LRIDTLDQIOAIHB 7.8 Ki 2
OFKKYVMUDLMESU 7.7 IC50 2
VQXSXVAWOWXDDK 7.7 Ki 2
ZBAAZUYUEZGUPA 7.7 Ki 2
VPTPOOCEAGWDJW 7.5 Ki 2
VZAFGXCWAWRULT 7.4 IC50 7
GUFVCUSKHSXTFY 7.4 IC50 2
CCSWDLQDJINVJP 7.3 Ki 2
OQXDWIBTIJGPGS 7.2 Ki 2
UXMGCZAWJOOQHZ 7.2 Ki 2
LIBRBDZWCDLREN 7.2 IC50 2
JYTISQGEFSHUIR 7.1 Kd 4
MSFPLTWUFWOKBX 7.1 IC50 2
PUFPGLSWMMJNSE 7.1 IC50 3
2D structure