Target Details
| UniProt AC | Q92830 |
|---|---|
| Gene Symbol | KAT2A |
| Protein Name | Histone acetyltransferase KAT2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00583 (Acetyltransf_1) PF00439 (Bromodomain) PF06466 (PCAF_N) |
Summary
- Multi-target molecules 55
- Clinical molecules 0
- Avg pChEMBL 8.54
KEGG Pathways (5)
Active Molecules (55)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVMOJFHRHLLSOT
|
6.8 | Kd | 3 | — | |
MSFPLTWUFWOKBX
|
6.7 | IC50 | 2 | — | |
XHAYAQCABOVSNX
|
6.6 | Kd | 9 | — | |
GVJYOLRRZZUUOE
|
6.4 | Kd | 5 | — | |
DBLNLPCEKQBLAI
|
6.3 | Kd | 3 | — |