Target Details
UniProt ACQ92830
Gene SymbolKAT2A
Protein NameHistone acetyltransferase KAT2A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00583 (Acetyltransf_1) PF00439 (Bromodomain) PF06466 (PCAF_N)
Summary
  • Multi-target molecules 55
  • Clinical molecules 0
  • Avg pChEMBL 8.54
Top Co-occurrence Targets
Active Molecules (55)
InChIKey pChEMBL Type Targets Clinical
MCIGDGJLNSNEHL 10.5 Ki 2
QSOFLSGOAZCHJA 10.3 Ki 2
TXWCNRCKXCEBOM 10.2 Ki 2
VMOQDLYJQCKIKJ 10.2 Ki 2
CPXKHLLAEZFPHJ 10.1 Ki 2
NOVLKEPNLVCXTE 10.0 Ki 2
FDEZYLHCNMEOEN 9.9 Ki 2
SCGIEXBRKPZTKA 9.9 Ki 2
ZKFBZQMNSFITPE 9.8 Ki 2
BWPNXWMSUALEOG 9.8 Ki 2
LRIDTLDQIOAIHB 9.8 Ki 2
ZMOIEFSZHIKKFS 9.7 Ki 2
NVXRVMGLQIHNFH 9.7 Ki 2
TVOCBMWTXJRBLB 9.6 Ki 2
RVZBXBUXJSRYKX 9.5 Ki 2
RJLFPNSUABSXRV 9.5 Ki 2
DBBDEGULRIBGMX 9.3 Ki 2
QOYJJEHJQBVOBM 9.3 Ki 2
UAIPDRJDVCRVGJ 9.3 Ki 2
CBPJBUBMKKGJMH 9.3 Ki 2
GXUCAUXOCJIOPD 9.2 Ki 2
SZITZWMQTGOBEC 9.1 Ki 2
VZAFGXCWAWRULT 8.9 Ki 7
KGYUNIZKDLZNSH 8.9 Ki 2
DAPYQEDLEDRHDE 8.9 Ki 2
ZWGAQZOUQSOIQA 8.8 Ki 2
LRIDTLDQIOAIHB 8.6 Ki 2
AXPLCJNXRWLGIP 8.5 Ki 2
SLWLRRQDEFXBSW 8.4 Ki 2
OZNYMBYLDCQTSZ 8.4 Ki 2
GJZNKOBWUOEFNR 8.3 Ki 2
NLMIRYVVKHZQBM 8.2 Ki 2
HINFIECYCWFNQN 8.2 Ki 2
YCXRPPJLAIUKFC 8.1 Ki 2
ZUUCCRLXECDZOE 8.0 Ki 2
ZBAAZUYUEZGUPA 8.0 Ki 2
OQXDWIBTIJGPGS 7.9 Ki 2
PYCNZAAZGQDRJG 7.9 IC50 2
CCSWDLQDJINVJP 7.8 Ki 2
VPTPOOCEAGWDJW 7.7 Ki 2
OFKKYVMUDLMESU 7.7 IC50 2
VQXSXVAWOWXDDK 7.7 Ki 2
HLMCIOPRABZQAU 7.5 Ki 2
FGVKACATFYZCMS 7.5 Ki 2
UXMGCZAWJOOQHZ 7.5 Ki 2
UOQAFGWMKNIVAR 7.4 Kd 6
JYTISQGEFSHUIR 7.2 Kd 4
LIBRBDZWCDLREN 7.2 IC50 2
PUFPGLSWMMJNSE 7.0 Kd 3
QFRIGJQJVRCBFQ 6.8 Kd 3
2D structure