Target Details
| UniProt AC | Q92824 |
|---|---|
| Gene Symbol | PCSK5 |
| Protein Name | Proprotein convertase subtilisin/kexin type 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14843 (GF_recep_IV) PF01483 (P_proprotein) PF00082 (Peptidase_S8) PF16470 (S8_pro-domain) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 7.21
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHBJTTGFHCHQHS
|
9.9 | Ki | 6 | — | |
RARQEZVPGNQDRL
|
8.8 | Ki | 5 | — | |
YGMAIAXBJLVVLI
|
8.8 | Ki | 5 | — | |
UXEFAKYOWKPLSZ
|
8.4 | Ki | 4 | — | |
YIMSHXFWBSXLKW
|
8.4 | Ki | 4 | — | |
CLTYJDDMFQEKEL
|
8.2 | Ki | 6 | — | |
QMAXHSLPLMYIPN
|
8.2 | Ki | 6 | — | |
ACPMDCNBPZRQGO
|
7.1 | Ki | 4 | — | |
HCRNWNCAUNWLJZ
|
7.1 | Ki | 4 | — | |
KWHYASXOKFJBKD
|
6.8 | Ki | 4 | — | |
LEEIZVYTIHJJNF
|
6.8 | Ki | 4 | — | |
GREDJTIKEQWSJW
|
6.7 | Ki | 4 | — | |
RYVHKZGUULZSGD
|
6.7 | Ki | 4 | — | |
CHSWXCHUJHYZLB
|
6.6 | Ki | 4 | — | |
XIHRZTWKTVFWSV
|
6.6 | Ki | 4 | — | |
ANHXASYJLDAVKI
|
6.4 | Ki | 4 | — | |
ALKYWGCWYLWWQX
|
6.3 | Ki | 4 | — | |
ICMPUUKPBRMOSD
|
6.3 | Ki | 4 | — | |
GBWNVGJPAAAKFV
|
6.2 | Ki | 3 | — | |
GHIUMDOROBFONL
|
6.2 | Ki | 3 | — | |
BEXKWEWEAXISEC
|
6.1 | Ki | 3 | — | |
SPILXWOFMWMUJL
|
6.1 | Ki | 3 | — |