Target Details
| UniProt AC | Q92800 |
|---|---|
| Gene Symbol | EZH1 |
| Protein Name | Histone-lysine N-methyltransferase EZH1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21358 (Ezh2_MCSS) PF11616 (EZH2_WD-Binding) PF18118 (PRC2_HTH_1) PF18264 (preSET_CXC) PF00856 (SET) |
Summary
- Multi-target molecules 65
- Clinical molecules 0
- Avg pChEMBL 7.68
KEGG Pathways (3)
Active Molecules (65)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKSFKBQGSFSOSM
|
6.9 | IC50 | 2 | — | |
AWROWLFZQZJJAH
|
6.9 | IC50 | 2 | — | |
NSQSAUGJQHDYNO
|
6.8 | IC50 | 6 | — | |
DEIZJPMLDLKNGP
|
6.8 | IC50 | 2 | — | |
CXLCYFIVMACFAK
|
6.8 | IC50 | 2 | — | |
LONVYJSHGSZBQY
|
6.8 | IC50 | 2 | — | |
ULNXAWLQFZMIHX
|
6.6 | IC50 | 7 | — | |
QKTOFXPWVLQIMX
|
6.5 | IC50 | 5 | — | |
KPLDMYFFSCWABC
|
6.4 | IC50 | 2 | — | |
QKZXBIXAKYLFRD
|
6.2 | IC50 | 2 | — | |
HRDQQHUKUIKFHT
|
6.2 | IC50 | 2 | — | |
RAHSOQYFNLKCMP
|
6.2 | IC50 | 2 | — | |
RNBZYKQPAMPZJW
|
6.1 | IC50 | 2 | — | |
SYBIETZSDORFFL
|
6.1 | IC50 | 2 | — | |
NQEWPBXAVVWIDZ
|
6.1 | IC50 | 2 | — |