Target Details
| UniProt AC | Q92794 |
|---|---|
| Gene Symbol | KAT6A |
| Protein Name | Histone acetyltransferase KAT6A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01853 (MOZ_SAS) PF00628 (PHD) PF21524 (SAMD1_WH) PF17772 (zf-MYST) |
Summary
- Multi-target molecules 359
- Clinical molecules 0
- Avg pChEMBL 7.87
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (359)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YEUSVVVKGKGBGT
|
7.3 | Ki | 3 | — | |
NWZKOEDRFSVGLU
|
7.3 | Ki | 2 | — | |
IQFYLVLGTKMSTF
|
7.3 | IC50 | 2 | — | |
DGDSIZMYTARPRE
|
7.3 | IC50 | 2 | — | |
FJXIXQMPONKCEK
|
7.3 | IC50 | 2 | — | |
MYXBTYIGTPOROK
|
7.2 | IC50 | 2 | — | |
AHUFEFPBCKDTPQ
|
7.2 | IC50 | 2 | — | |
XKBVDFIVHCHXTG
|
7.2 | IC50 | 2 | — | |
YCKKFNVIWHRJIL
|
7.2 | IC50 | 2 | — | |
WUFJYHONWVWZBJ
|
7.2 | Ki | 2 | — | |
FZKNVOUHIRQWIZ
|
7.2 | IC50 | 2 | — | |
GOQGPSRYBRCOHR
|
7.2 | Ki | 2 | — | |
DAAVLQGOUKVRQI
|
7.2 | IC50 | 2 | — | |
HDLLRNNSKMPHDD
|
7.2 | Ki | 2 | — | |
RPNBGMRKQRNGOA
|
7.2 | IC50 | 2 | — | |
YYUSTIDFVBSASR
|
7.2 | IC50 | 2 | — | |
AROLCXGYORHJGB
|
7.2 | IC50 | 2 | — | |
WWFRXLVYYYMFTR
|
7.2 | Ki | 2 | — | |
ILZSLOIWTWYVKB
|
7.2 | IC50 | 3 | — | |
RZWDESKLSMUQIH
|
7.2 | Ki | 2 | — | |
VNQYVJVOOYJXTE
|
7.2 | IC50 | 2 | — | |
UKUDAABFNFVXKZ
|
7.2 | IC50 | 2 | — | |
MDCIIHVXSGUGGI
|
7.1 | IC50 | 2 | — | |
RLVDXRFINQZHHI
|
7.1 | IC50 | 2 | — | |
MUDWLAWEYKBEKT
|
7.1 | IC50 | 2 | — | |
ZVOLLEIEPYCTPO
|
7.1 | IC50 | 2 | — | |
FVTNUOYDCMTVJV
|
7.1 | IC50 | 2 | — | |
LLOVJXVFXXQLAT
|
7.1 | IC50 | 2 | — | |
XUTASFIPHCWYFX
|
7.1 | IC50 | 2 | — | |
JYEYJYMNQVNPQV
|
7.1 | IC50 | 2 | — | |
KLISXWOCRBBTDK
|
7.1 | IC50 | 2 | — | |
JFFDRYBVVLPPHL
|
7.1 | IC50 | 2 | — | |
ZUWIDJYXRPTMQW
|
7.1 | IC50 | 2 | — | |
ZPSLBWHEMLEUDR
|
7.0 | IC50 | 2 | — | |
OBLBXCVBYBHIOD
|
7.0 | Ki | 3 | — | |
WSOJKPLHXJCURO
|
7.0 | IC50 | 2 | — | |
RKUWEXNFEXZQMX
|
7.0 | IC50 | 2 | — | |
BXSNCLQDVZAUQY
|
7.0 | IC50 | 2 | — | |
STYLGRNBUZFUJF
|
7.0 | Ki | 3 | — | |
FPZFQKIBPOZLHQ
|
7.0 | IC50 | 2 | — | |
SUZNSHMEVWQFIQ
|
7.0 | IC50 | 2 | — | |
VJEHDXGZSHZNHT
|
7.0 | IC50 | 2 | — | |
SNBRNUWZDKKREE
|
7.0 | IC50 | 2 | — | |
CEHZZQQQSCOXRQ
|
7.0 | IC50 | 2 | — | |
KMQMZYHNMLFPAF
|
7.0 | IC50 | 2 | — | |
UFZNEGKLNAWKQR
|
7.0 | IC50 | 2 | — | |
CQQDHHNIZBAZFB
|
7.0 | Ki | 2 | — | |
QIQSSWVSUWKSLY
|
7.0 | IC50 | 2 | — | |
DUQUVGVUEONHMM
|
6.9 | IC50 | 2 | — | |
IHZUSHOOBNVREF
|
6.9 | IC50 | 2 | — |