Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GVSZNXQDVTYYAN
|
6.5 | IC50 | 2 | — | |
SRFOIWNXIILSNJ
|
6.5 | IC50 | 4 | — | |
ZHMCGBRGDVCXLS
|
6.5 | IC50 | 5 | — | |
NPKBSQHTYBKPJD
|
6.5 | IC50 | 2 | — | |
QWJMFUIHTVAUCH
|
6.5 | IC50 | 3 | — | |
ZOVYOHAZPIKVOR
|
6.5 | IC50 | 4 | — | |
BMBTWLMYKIAXLA
|
6.5 | IC50 | 2 | — | |
HJDWUDBQIKJSJE
|
6.5 | Kd | 2 | — | |
UWQPEIABRDXMTQ
|
6.5 | IC50 | 2 | — | |
ZVYCZICBBIUVHC
|
6.5 | Kd | 3 | — | |
FBGWKDHQIRVFSD
|
6.5 | IC50 | 2 | — | |
RONQAYQWPFKHGK
|
6.5 | IC50 | 2 | — | |
WNTOXMAGPDYDCR
|
6.5 | IC50 | 3 | — | |
KECYVMVFYPBARC
|
6.5 | IC50 | 2 | — | |
OTLUGLDCVHKZEE
|
6.5 | IC50 | 2 | — | |
FMFGVLUVPAHDDT
|
6.5 | IC50 | 2 | — | |
ICKGOXSYBTWKAP
|
6.5 | IC50 | 2 | — | |
LPWRLICNAUJRIQ
|
6.5 | IC50 | 2 | — | |
UUBWOQFEIRJDKR
|
6.5 | IC50 | 2 | — | |
RPOVNYLBJCXTOQ
|
6.5 | IC50 | 2 | — | |
ICGXDGBYQZIXIF
|
6.5 | IC50 | 2 | — | |
ZHQPTIFREKVURJ
|
6.5 | IC50 | 2 | — | |
CUQCNMCZQPPDII
|
6.4 | IC50 | 2 | — | |
WQRKDXUDKMFKPL
|
6.4 | IC50 | 4 | — | |
XSISVIBLCIAEGR
|
6.4 | IC50 | 4 | — | |
BKOMFGNROQEUHF
|
6.4 | IC50 | 2 | — | |
IVXYIGADMWHQDD
|
6.4 | IC50 | 4 | — | |
CUAGRANTRNSGSF
|
6.4 | IC50 | 2 | — | |
GAFYFVRFEKFZOU
|
6.4 | IC50 | 4 | — | |
OPRLJTKXGDBVAC
|
6.4 | IC50 | 2 | — | |
OYPQYGXUQANMSS
|
6.4 | IC50 | 2 | — | |
DGJREYHVQYZTEV
|
6.4 | Kd | 6 | — | |
RJCJQUKBDBNIOB
|
6.4 | IC50 | 4 | — | |
OSOMHZBGIZCTKM
|
6.4 | IC50 | 4 | — | |
XMANXVDMULPMRR
|
6.4 | IC50 | 2 | — | |
ZTGCZUISBHLGKD
|
6.4 | IC50 | 2 | — | |
PWPYJSVOLAVRNB
|
6.4 | IC50 | 2 | — | |
OGSOMZCUMMDDJU
|
6.3 | IC50 | 4 | — | |
IMXDUOIANVGJIA
|
6.3 | IC50 | 4 | — | |
HPSNXSAYALRMQW
|
6.3 | IC50 | 2 | — | |
UQMYMWRETIHSGQ
|
6.3 | IC50 | 3 | — | |
PJFBYCXYSAXHLS
|
6.3 | IC50 | 2 | — | |
VBRWZRVQWASOOS
|
6.3 | IC50 | 2 | — | |
ZGPUZLWYKXAJNB
|
6.3 | IC50 | 2 | — | |
KSYAZQGGEUUIPO
|
6.3 | IC50 | 2 | — | |
LCYKVOFPEMZEDI
|
6.3 | IC50 | 2 | — | |
SDLMPYCGZKLARA
|
6.3 | IC50 | 4 | — | |
WIXBOVBNLLVASA
|
6.3 | IC50 | 2 | — | |
AEANZCXROGPSBY
|
6.3 | Kd | 6 | — | |
FMTAQWMOLHFOLT
|
6.3 | Kd | 2 | — |