Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PWOWVSPUJRPEGX
|
6.8 | IC50 | 2 | — | |
GMINUTRRQLVDKN
|
6.8 | IC50 | 2 | — | |
LGSNHFDNKYQHEI
|
6.8 | IC50 | 2 | — | |
OPRLJTKXGDBVAC
|
6.8 | IC50 | 2 | — | |
RAIPQLGDNRXVJX
|
6.8 | IC50 | 2 | — | |
ICUFVYYLUGJQPU
|
6.8 | IC50 | 2 | — | |
NGRKNMYUPWAPCQ
|
6.8 | IC50 | 2 | — | |
KHQQNXFBTALTQF
|
6.8 | Kd | 6 | — | |
YKNAKDFZAWQEEO
|
6.8 | Kd | 3 | — | |
FAZFZYDAOJWKSE
|
6.8 | IC50 | 2 | — | |
PEYCCFBAPYGGOX
|
6.8 | IC50 | 2 | — | |
SNLNRCQNXQMLNB
|
6.8 | IC50 | 2 | — | |
UWZMEPZRQVYBCI
|
6.8 | IC50 | 2 | — | |
YWMBZVKDVIDBAQ
|
6.8 | IC50 | 2 | — | |
NFMDDLDYDOZPGW
|
6.8 | IC50 | 2 | — | |
CEPJZYYWEDIEOG
|
6.7 | IC50 | 2 | — | |
XSOFZNARGSJIQN
|
6.7 | IC50 | 4 | — | |
HSOYPKXYVCVZOK
|
6.7 | IC50 | 2 | — | |
RZNVPBJTIYRMSE
|
6.7 | IC50 | 2 | — | |
RZYSZTUMZFCLCL
|
6.7 | IC50 | 2 | — | |
XNMUDJLUIVAEFS
|
6.7 | IC50 | 2 | — | |
HPXHQNWBKFNTMR
|
6.7 | IC50 | 2 | — | |
QCVBUWRWHOLCOJ
|
6.7 | IC50 | 2 | — | |
IMLLQTJDJJVPOT
|
6.7 | IC50 | 2 | — | |
WLUMGCPGWDQOSB
|
6.7 | IC50 | 3 | — | |
DKCFKYUXDNTZAE
|
6.7 | IC50 | 2 | — | |
IFFAPYISKKZOPO
|
6.7 | IC50 | 4 | — | |
ZSTNBLSPAMZIQD
|
6.7 | IC50 | 2 | — | |
ZUDONVCZBCQPST
|
6.7 | IC50 | 2 | — | |
YPPIBRNYHDEWID
|
6.7 | IC50 | 2 | — | |
NZAWVJDDBLNIQI
|
6.7 | IC50 | 2 | — | |
OEKXMLFJULWEJI
|
6.7 | Kd | 2 | — | |
FEVFEDHOYMRQIZ
|
6.6 | IC50 | 2 | — | |
JQHRYVMEBZSFGK
|
6.6 | Kd | 2 | — | |
FQVGCUZGXCCGOC
|
6.6 | IC50 | 2 | — | |
LVVCZEJBVPEPGJ
|
6.6 | IC50 | 2 | — | |
NYYPYDLZLGCKOU
|
6.6 | IC50 | 4 | — | |
LXEXKNGUTAFYKW
|
6.6 | IC50 | 2 | — | |
NWIFMQIVWVMZLD
|
6.6 | IC50 | 2 | — | |
BQDONWPMBNKZCG
|
6.6 | IC50 | 4 | — | |
BVNSMRUDPSJEIU
|
6.6 | IC50 | 2 | — | |
ISWOCAVPQAAWOZ
|
6.6 | IC50 | 2 | — | |
UGVSWFJGRKHVMD
|
6.6 | IC50 | 4 | — | |
LVVCZEJBVPEPGJ
|
6.5 | IC50 | 2 | — | |
RGKUFEQXYKVMOO
|
6.5 | IC50 | 4 | — | |
BPKDBMDIWIBGMA
|
6.5 | IC50 | 2 | — | |
OJPOVVTUDJNUND
|
6.5 | IC50 | 2 | — | |
RKCDVGZWRITJMS
|
6.5 | IC50 | 2 | — | |
ARBRHWRTXPWZGN
|
6.5 | IC50 | 5 | — | |
DREXABSQFKJHIP
|
6.5 | IC50 | 2 | — |