Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QAMFZTLDTZXWMB
|
7.3 | IC50 | 2 | — | |
QIEZNDCYIUHVBH
|
7.3 | IC50 | 2 | — | |
RBTJDFWZAROJPI
|
7.3 | IC50 | 2 | — | |
RDAUNHLHLBFFIG
|
7.3 | IC50 | 2 | — | |
RSPLKXLEIPCXMI
|
7.3 | IC50 | 2 | — | |
SHJSPBYADHRCRL
|
7.3 | IC50 | 2 | — | |
SLWYCOVLGHZAFK
|
7.3 | IC50 | 2 | — | |
VPYWJZXADHWXKN
|
7.3 | IC50 | 2 | — | |
VQQUAHKOKFMQNX
|
7.3 | IC50 | 2 | — | |
WBRLENDDMAMVNQ
|
7.3 | IC50 | 2 | — | |
WNRPGGJJNZESRC
|
7.3 | IC50 | 2 | — | |
WOLOIHALMNZHJK
|
7.3 | IC50 | 2 | — | |
XLBMIRHNQUWVAM
|
7.3 | IC50 | 2 | — | |
XOJFGGXGCDNCQP
|
7.3 | IC50 | 2 | — | |
ZECXHJZIVFQVHV
|
7.3 | IC50 | 2 | — | |
ZOHWOLKQTZMORA
|
7.3 | IC50 | 2 | — | |
ZYXKYFZBMMBZJZ
|
7.3 | IC50 | 2 | — | |
VVOJECSTVKGBLZ
|
7.2 | IC50 | 3 | — | |
QKJJFWYEGUSNLI
|
7.2 | IC50 | 2 | — | |
RGAAGDNMRXFIBD
|
7.2 | IC50 | 2 | — | |
RFOWAAZLTHLZHO
|
7.1 | IC50 | 2 | — | |
HMMXTPNGIWNLQA
|
7.1 | IC50 | 2 | — | |
QEBQWMOQSWEYPS
|
7.1 | IC50 | 2 | — | |
RWUFFMJUVGICHP
|
7.1 | IC50 | 2 | — | |
LDPBOBQZOFLMLU
|
7.1 | IC50 | 3 | — | |
RCPJEOKKJODBRQ
|
7.1 | IC50 | 2 | — | |
XVPFIRFAOOSQTK
|
7.1 | IC50 | 2 | — | |
KAGYLLHUHGBNTA
|
7.0 | IC50 | 2 | — | |
QLRYSHYUZMZZPY
|
7.0 | IC50 | 4 | — | |
XUGFYFHLYOPQJS
|
7.0 | IC50 | 2 | — | |
BAHQNJLZVVLSJW
|
7.0 | IC50 | 2 | — | |
PMNZVZQYPSMXDO
|
7.0 | IC50 | 2 | — | |
WSOSPNZDGBUARC
|
7.0 | IC50 | 2 | — | |
VBTDHMQUNCGCSZ
|
7.0 | Kd | 2 | — | |
UOGTVNXJONPDSD
|
7.0 | IC50 | 2 | — | |
FTTXUZIHQYKOBF
|
7.0 | IC50 | 2 | — | |
LMLIBNUOIWAJFC
|
7.0 | Kd | 9 | — | |
PSFDBOWKEFILAQ
|
7.0 | IC50 | 2 | — | |
RQFUKBAHMUVXDA
|
6.9 | IC50 | 2 | — | |
ZNIQPKLUCOYTFF
|
6.9 | IC50 | 2 | — | |
LPEFXYUIOKMUCW
|
6.9 | IC50 | 2 | — | |
CGWBJJZOKGZCSJ
|
6.9 | IC50 | 3 | — | |
QQUFYDKFQLICRA
|
6.9 | IC50 | 2 | — | |
WQEGQSRMXSLEON
|
6.9 | IC50 | 4 | — | |
PSWWDDSOCOGNCT
|
6.9 | IC50 | 2 | — | |
CUJLWYCUPPPASA
|
6.9 | Kd | 2 | — | |
QESLMEPTLHITHH
|
6.9 | IC50 | 2 | — | |
LQUIXMWIBNXAAR
|
6.8 | IC50 | 2 | — | |
NZXSWCLCRDCHGN
|
6.8 | IC50 | 2 | — | |
VHOZWHQPEJGPCC
|
6.8 | IC50 | 3 | — |