Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BHFMWVNKVQLZBG
|
7.4 | Kd | 2 | — | |
IQDDINKYXBDMEA
|
7.4 | IC50 | 2 | — | |
SGNUOADKIKQBIW
|
7.4 | IC50 | 2 | — | |
ANIBATUKYBCBNA
|
7.4 | IC50 | 2 | — | |
IKUNJTRUFVIYTB
|
7.4 | IC50 | 2 | — | |
NKOJNOBJGYTLLZ
|
7.4 | IC50 | 2 | — | |
NSRRDNGMQXSHPJ
|
7.4 | IC50 | 2 | — | |
SSTRQKVGFZOZCS
|
7.4 | IC50 | 2 | — | |
VWZAAFMUYDNGED
|
7.4 | IC50 | 2 | — | |
UYFJLWOWNNRESN
|
7.4 | IC50 | 2 | — | |
QHEXIHFMBFZCSJ
|
7.4 | IC50 | 2 | — | |
JIYPVUCBRQNICX
|
7.3 | Kd | 7 | — | |
DJNGAENPUAKERE
|
7.3 | IC50 | 2 | — | |
JGAVEEORSJOUOB
|
7.3 | IC50 | 2 | — | |
AORCBCMGWOSZPF
|
7.3 | IC50 | 2 | — | |
BBVMUXYYTMWPPB
|
7.3 | IC50 | 2 | — | |
BLYPILQXQHVPJW
|
7.3 | IC50 | 2 | — | |
CCEZKQROHBLKNL
|
7.3 | IC50 | 2 | — | |
CFUIPJIOBHPOKQ
|
7.3 | IC50 | 2 | — | |
CXWTZSOLFHGXRT
|
7.3 | IC50 | 2 | — | |
DMHBFVKGGJRPSC
|
7.3 | IC50 | 2 | — | |
DZILMUATPGLNCF
|
7.3 | IC50 | 2 | — | |
FMMFNIRCAYUISW
|
7.3 | IC50 | 2 | — | |
FPEGMSVGVYBBLT
|
7.3 | IC50 | 2 | — | |
FTEKTWXFBITADQ
|
7.3 | IC50 | 2 | — | |
GDTRZUHBRQHCKF
|
7.3 | IC50 | 2 | — | |
GFPXDXYANNOFDI
|
7.3 | IC50 | 2 | — | |
GNPKTOPHGVBHCK
|
7.3 | IC50 | 2 | — | |
HTSHGKTUFLVKOK
|
7.3 | IC50 | 2 | — | |
ICEINJFBCBLFQW
|
7.3 | IC50 | 2 | — | |
IIBPTHUAQTYNPQ
|
7.3 | IC50 | 2 | — | |
IOLAIYBRDIUGFO
|
7.3 | IC50 | 2 | — | |
IRMYWCSBRPICRR
|
7.3 | IC50 | 2 | — | |
ITIJQWPCABXZNE
|
7.3 | IC50 | 2 | — | |
IYBQCTFBCWEMNR
|
7.3 | IC50 | 2 | — | |
JGIORIYESNLPAE
|
7.3 | IC50 | 2 | — | |
JQKFQKWNJCVSKS
|
7.3 | IC50 | 2 | — | |
JWSSFNCIAIVAQB
|
7.3 | IC50 | 2 | — | |
KMMRUIFQVRRCDS
|
7.3 | IC50 | 2 | — | |
KQPLCOWNYYXDDH
|
7.3 | IC50 | 2 | — | |
LCWFKXOJTKLMHT
|
7.3 | IC50 | 2 | — | |
LOKYREGDIHEAIW
|
7.3 | IC50 | 2 | — | |
MSCMIRSJVCNMNP
|
7.3 | IC50 | 2 | — | |
MWVOGVAMNZFYGO
|
7.3 | IC50 | 2 | — | |
MWWTYIJAMGUEKI
|
7.3 | IC50 | 2 | — | |
NMVOEOLFZMQWNV
|
7.3 | IC50 | 2 | — | |
NZDVOYUYYDTMAH
|
7.3 | IC50 | 2 | — | |
OCIHEXBMLNGWJE
|
7.3 | IC50 | 2 | — | |
PIOSPEYIKUSPGY
|
7.3 | IC50 | 2 | — | |
PPJFPDJMQHNWPW
|
7.3 | IC50 | 2 | — |