Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KBMLUWNAWHJXMZ
|
7.8 | IC50 | 2 | — | |
MTRFXIUYTHPDTC
|
7.8 | IC50 | 2 | — | |
NJVMBNYLGJNKFJ
|
7.8 | IC50 | 2 | — | |
NOUKMOKAEKAWKS
|
7.8 | IC50 | 2 | — | |
OEOQBFZBBBRFIS
|
7.8 | IC50 | 2 | — | |
RJGAUFFLIIPBSF
|
7.8 | IC50 | 2 | — | |
SSODXDQRZAFRQH
|
7.8 | IC50 | 2 | — | |
UWPPBQXHMIAQRE
|
7.8 | IC50 | 2 | — | |
VJBQAWIJVMWZBJ
|
7.8 | IC50 | 2 | — | |
VKFMVPDPCOIPQY
|
7.8 | IC50 | 2 | — | |
WMCRMAIKKKCSMD
|
7.8 | IC50 | 2 | — | |
XAKNSTLMMUROQR
|
7.8 | IC50 | 2 | — | |
YJSOMEGWZGMTKF
|
7.8 | IC50 | 2 | — | |
YWHJHAFMEISKFY
|
7.8 | IC50 | 2 | — | |
XIRSITKWZXVEPU
|
7.7 | Kd | 2 | — | |
YGZKIOPJGFQDSR
|
7.7 | Ki | 2 | — | |
IFIMPCBCWYNSEK
|
7.7 | IC50 | 2 | — | |
MKHZYJVBJCVUJD
|
7.7 | IC50 | 3 | — | |
OMECDPIDDYPFQD
|
7.7 | IC50 | 2 | — | |
SVADXQXVQIZUOT
|
7.7 | IC50 | 3 | — | |
IQZLAXNGIATBBF
|
7.7 | IC50 | 3 | — | |
KPWWFNXRLAAREN
|
7.7 | Kd | 12 | — | |
LVZJYBDBJTYEPA
|
7.7 | Kd | 2 | — | |
OQHPHGZWSTYMIQ
|
7.7 | IC50 | 3 | — | |
JPEYACZELJYCMI
|
7.7 | IC50 | 2 | — | |
WNMRBAPHMQERLK
|
7.7 | Kd | 2 | — | |
NOKDEWTXUBQOFY
|
7.6 | IC50 | 2 | — | |
LJIYNYPVUBPNRT
|
7.6 | IC50 | 2 | — | |
VLSSRXAUNKQKKE
|
7.6 | IC50 | 2 | — | |
BMFWCARUVZTJGG
|
7.5 | Kd | 2 | — | |
DBCMAPQJHUHFJH
|
7.5 | IC50 | 2 | — | |
VDINOEOOUILKFN
|
7.5 | IC50 | 2 | — | |
GEPYBHCJBORHCE
|
7.5 | IC50 | 3 | — | |
AMNYDJDEGBTNSA
|
7.5 | IC50 | 2 | — | |
BFTKDWYIRJGJCA
|
7.5 | IC50 | 3 | — | |
HLTFLEHNLNKZIT
|
7.5 | IC50 | 2 | — | |
JYEGHZZFDPRSDT
|
7.5 | IC50 | 2 | — | |
KDQSAWDSOXZXES
|
7.5 | IC50 | 2 | — | |
NPRLPBVOWPMZCP
|
7.5 | IC50 | 2 | — | |
QFOWHCHCRRILAW
|
7.5 | IC50 | 2 | — | |
WYXLFFVUWVUYOG
|
7.5 | Kd | 2 | — | |
YHBKXFFZZJCTSD
|
7.5 | IC50 | 2 | — | |
YSBDLHAKVVSCMY
|
7.5 | IC50 | 2 | — | |
ZDLOIRATYRBXGM
|
7.5 | IC50 | 2 | — | |
ZNIQPKLUCOYTFF
|
7.5 | IC50 | 2 | — | |
UXTBGAAKAKILOF
|
7.5 | Kd | 2 | — | |
YNLJURILQNEPQG
|
7.5 | Kd | 2 | — | |
DREXABSQFKJHIP
|
7.5 | IC50 | 2 | — | |
FQVXPGXSEMNATG
|
7.4 | IC50 | 2 | — | |
JTGDKTAYORPKNS
|
7.4 | Kd | 2 | — |