Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PGHWEDXBYGEVHA
|
8.3 | IC50 | 2 | — | |
PPXPAULWKFUZOS
|
8.3 | IC50 | 2 | — | |
PTMNXXOEXDHJJZ
|
8.3 | IC50 | 2 | — | |
QGGTYOVAUVANML
|
8.3 | IC50 | 2 | — | |
QGGVBTFIDGXVTH
|
8.3 | IC50 | 2 | — | |
QSKCPIMTMWXKEN
|
8.3 | IC50 | 2 | — | |
RGEYHNPTYRAWSW
|
8.3 | IC50 | 2 | — | |
RVWUEZKBPVHOOY
|
8.3 | IC50 | 2 | — | |
RZSYDFQOGZBKKB
|
8.3 | IC50 | 2 | — | |
SFYVTHBCERVFDA
|
8.3 | IC50 | 2 | — | |
SOLDGMQYVHLMIE
|
8.3 | IC50 | 2 | — | |
SQXQLPYRXYYOBM
|
8.3 | IC50 | 2 | — | |
SWHRRNMZQZWREJ
|
8.3 | IC50 | 2 | — | |
TZBNCXYMRLRVFB
|
8.3 | IC50 | 2 | — | |
UAPROUKGMPFZNW
|
8.3 | IC50 | 2 | — | |
UCFSUNZUUXRHAH
|
8.3 | IC50 | 2 | — | |
UFYXPMMBZOBVAH
|
8.3 | IC50 | 2 | — | |
VSXZMQRFGTUJQG
|
8.3 | IC50 | 2 | — | |
WOJQJMZZSQTUFQ
|
8.3 | IC50 | 2 | — | |
WQNHOBLKGYIXPH
|
8.3 | IC50 | 2 | — | |
XTDSIZPENIOUII
|
8.3 | IC50 | 2 | — | |
XVKVQNMVFBUYCC
|
8.3 | IC50 | 2 | — | |
YIHSGBIQASYBCF
|
8.3 | IC50 | 2 | — | |
YLKGVDDJDVHJHR
|
8.3 | IC50 | 2 | — | |
YROQFFIYPKVCOA
|
8.3 | IC50 | 2 | — | |
YYJXCCVGEHXJBS
|
8.3 | IC50 | 2 | — | |
ZJGMOHOOSGHFMJ
|
8.2 | IC50 | 2 | — | |
GNHYVESLYMWXEL
|
8.2 | IC50 | 2 | — | |
YXSUJYIAFJZLAJ
|
8.2 | IC50 | 2 | — | |
GGXPWHYWZIJKLJ
|
8.1 | IC50 | 2 | — | |
QULMQLITKMCMAK
|
8.1 | IC50 | 2 | — | |
COHJFFNOXQFYOA
|
8.0 | IC50 | 2 | — | |
FNFTWNFLHHXYIF
|
8.0 | IC50 | 2 | — | |
NRROGCBXQIAIEQ
|
8.0 | IC50 | 2 | — | |
RYCIBPVLRWPLSI
|
8.0 | IC50 | 2 | — | |
XDPSVWUCEHLIOX
|
8.0 | IC50 | 2 | — | |
ATLJVYAAMGQNOV
|
7.9 | IC50 | 2 | — | |
VRVJKILQRBSEAG
|
7.9 | IC50 | 3 | — | |
OLGHKQPFBIYQAO
|
7.8 | IC50 | 2 | — | |
KKCORLIQMAQULG
|
7.8 | IC50 | 2 | — | |
BQHGAFARPXXMCN
|
7.8 | IC50 | 2 | — | |
DJGKXQJOJGSFCC
|
7.8 | IC50 | 2 | — | |
DNOQGYIZSIKUKV
|
7.8 | IC50 | 2 | — | |
FKUZJBDMRFPBGZ
|
7.8 | IC50 | 2 | — | |
FPEUVFGHEOYIEY
|
7.8 | IC50 | 2 | — | |
GQBOHKSNHSHUAO
|
7.8 | IC50 | 2 | — | |
GZRGMPOBPUOPHW
|
7.8 | IC50 | 2 | — | |
HWOWLOFMYRGPGJ
|
7.8 | IC50 | 2 | — | |
HYGYLJIDGVHEBB
|
7.8 | IC50 | 2 | — | |
IGNITTXLQQFMPB
|
7.8 | IC50 | 2 | — |