Target Details
| UniProt AC | Q92793 |
|---|---|
| Gene Symbol | CREBBP |
| Protein Name | CREB-binding protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF09030 (Creb_binding) PF08214 (HAT_KAT11) PF02172 (KIX) PF23570 (PHD_P300) PF06001 (RING_CBP-p300) PF02135 (zf-TAZ) PF00569 (ZZ) |
Summary
- Multi-target molecules 423
- Clinical molecules 0
- Avg pChEMBL 7.16
KEGG Pathways (29)
- Adherens junction
- Cadherin signaling
- Cell cycle
- FoxO signaling pathway
- Glucagon signaling pathway
- Growth hormone synthesis, secretion and action
- HIF-1 signaling pathway
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Huntington disease
- Influenza A
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Long-term potentiation
- Melanogenesis
- MicroRNAs in cancer
- Notch signaling pathway
- Pathways in cancer
- Polycomb repressive complex
- Prostate cancer
- Renal cell carcinoma
- TGF-beta signaling pathway
- Thyroid hormone signaling pathway
- Tuberculosis
- Viral carcinogenesis
- Viral life cycle - HIV-1
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPCJDXNTSDAQDE
|
9.2 | IC50 | 2 | — | |
OISTZKLYQBJTIE
|
9.2 | IC50 | 2 | — | |
MUJXZEDIWKGKQD
|
9.0 | IC50 | 2 | — | |
UCKDTCZSOLMOMQ
|
9.0 | IC50 | 2 | — | |
SKDNDJWEBPQKCS
|
8.8 | Kd | 3 | — | |
SKDNDJWEBPQKCS
|
8.6 | IC50 | 5 | — | |
VRVJKILQRBSEAG
|
8.6 | IC50 | 2 | — | |
SEDFZSHSBUXKAC
|
8.5 | IC50 | 2 | — | |
MSDYJZMQGKWYMG
|
8.5 | IC50 | 2 | — | |
ZEMJUJNMCGYHGO
|
8.5 | IC50 | 3 | — | |
AOJQXLVQLJFNQK
|
8.3 | IC50 | 2 | — | |
ARVSOFZRHJPWRD
|
8.3 | IC50 | 2 | — | |
BAMVRCOHSWSONB
|
8.3 | IC50 | 2 | — | |
BRSZRELKDMVWLF
|
8.3 | IC50 | 2 | — | |
CDDHJCJHOGVCQL
|
8.3 | IC50 | 2 | — | |
CHPASXRQUZTLJV
|
8.3 | IC50 | 2 | — | |
CHPASXRQUZTLJV
|
8.3 | IC50 | 2 | — | |
CNKPKJKOYIATHW
|
8.3 | IC50 | 2 | — | |
CNKPKJKOYIATHW
|
8.3 | IC50 | 2 | — | |
CRFKDPLPAGNYNW
|
8.3 | IC50 | 2 | — | |
CTFVIJXSVJYDGH
|
8.3 | IC50 | 2 | — | |
CUZFYOMNIRBZGO
|
8.3 | IC50 | 2 | — | |
DILBTBIYEGCJDD
|
8.3 | IC50 | 2 | — | |
DMHBFVKGGJRPSC
|
8.3 | IC50 | 2 | — | |
FMAIZEHZDPUEJB
|
8.3 | IC50 | 2 | — | |
GALGGCVHDILEOG
|
8.3 | IC50 | 2 | — | |
HOGUTLRARYUPKE
|
8.3 | IC50 | 2 | — | |
IJHCMDLIRJQLFI
|
8.3 | IC50 | 2 | — | |
IMEZXBOKDHUIFH
|
8.3 | IC50 | 2 | — | |
IUSALJIMSCCGFF
|
8.3 | IC50 | 2 | — | |
IXPPCILHCIJIID
|
8.3 | IC50 | 2 | — | |
JKKQEUVAOJAFJX
|
8.3 | IC50 | 2 | — | |
JVIJCKATFNYBOD
|
8.3 | IC50 | 2 | — | |
KIHKNKIFDMAUKT
|
8.3 | IC50 | 2 | — | |
KLKJKELOLLNBJQ
|
8.3 | IC50 | 2 | — | |
KNZBWHGOKBRMKI
|
8.3 | IC50 | 2 | — | |
KZSGWGCOCZVNRL
|
8.3 | IC50 | 2 | — | |
KZWWSHDZYVYUEX
|
8.3 | IC50 | 2 | — | |
LDMLSHJWWCAVGO
|
8.3 | IC50 | 2 | — | |
LFXSAVRBMNETDK
|
8.3 | IC50 | 2 | — | |
LGJNYOLMCOQCOZ
|
8.3 | IC50 | 2 | — | |
LNWUHDLNKXMJNO
|
8.3 | IC50 | 2 | — | |
LRBBMCOGXASSSU
|
8.3 | IC50 | 2 | — | |
LZDQOYFBIASSKS
|
8.3 | IC50 | 2 | — | |
MFLZAZRVKSCKAY
|
8.3 | IC50 | 2 | — | |
MOHNOQZUOQAGGB
|
8.3 | IC50 | 2 | — | |
NCWBIBOIJCSXLK
|
8.3 | IC50 | 2 | — | |
NSASXGLSRRHMCJ
|
8.3 | IC50 | 2 | — | |
OPLLJRZYXODUEK
|
8.3 | IC50 | 2 | — | |
OTKHTWOKGSLJOV
|
8.3 | IC50 | 2 | — |