Target Details
| UniProt AC | Q92772 |
|---|---|
| Gene Symbol | CDKL2 |
| Protein Name | Cyclin-dependent kinase-like 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 18
- Clinical molecules 7
- Avg pChEMBL 6.76
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODPGGGTTYSGTGO
|
9.3 | Kd | 153 | — | |
OUSFTKFNBAZUKL
|
7.4 | Kd | 58 | Yes | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
GCIKSSRWRFVXBI
|
7.3 | Kd | 109 | Yes | |
MLDQJTXFUGDVEO
|
6.9 | Kd | 85 | Yes | |
ASGMFNBUXDJWJJ
|
6.8 | IC50 | 8 | — | |
PIQCTGMSNWUMAF
|
6.7 | Kd | 137 | Yes | |
IIKPYJZUOZRTIB
|
6.6 | IC50 | 4 | — | |
CXQHYVUVSFXTMY
|
6.6 | Kd | 154 | — | |
JSAQBOQCZJHWMA
|
6.6 | Kd | 11 | — | |
SEJGTFPOEJWEGG
|
6.6 | Kd | 149 | — | |
BMWMKGNVAMXXCH
|
6.4 | Kd | 6 | — | |
HKSZLNNOFSGOKW
|
6.3 | Kd | 408 | — | |
RITAVMQDGBJQJZ
|
6.3 | Kd | 43 | — | |
DPCPNRYPXUUJCP
|
6.3 | IC50 | 4 | — | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
UCBIQZUJJSVQHL
|
6.1 | Kd | 8 | — | |
OVPNQJVDAFNBDN
|
6.0 | Kd | 44 | Yes |