Target Details
| UniProt AC | Q92633 |
|---|---|
| Gene Symbol | LPAR1 |
| Protein Name | Lysophosphatidic acid receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 122
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (8)
Active Molecules (122)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SKDIMRRKRVTENP
|
6.7 | IC50 | 2 | — | |
AKIUAYSBXDBMOX
|
6.6 | IC50 | 2 | — | |
XHZMTTZICDAOHN
|
6.5 | IC50 | 2 | — | |
XYSBQYUENLDGMI
|
6.5 | IC50 | 2 | — | |
WFNXESYFHAMZSY
|
6.5 | Ki | 2 | — | |
SQFNSQHVILJRSM
|
6.4 | IC50 | 2 | — | |
NSVGYWDUGKCWRF
|
6.4 | IC50 | 2 | — | |
ONGMIZHEZHGEOT
|
6.3 | IC50 | 2 | — | |
VKPRWVOYFUXFAT
|
6.3 | Ki | 2 | — | |
LLIFMNUXGDHTRO
|
6.3 | IC50 | 2 | — | |
VNBIUEOBRLCNQI
|
6.3 | IC50 | 2 | — | |
GDLXQEKNJMCXRS
|
6.3 | Ki | 2 | — | |
CUXSKJSPPDINEH
|
6.3 | IC50 | 3 | — | |
XYSBQYUENLDGMI
|
6.3 | IC50 | 2 | — | |
TXROCRKOYMGIGD
|
6.3 | IC50 | 2 | — | |
YZILIQNNTIKUCA
|
6.2 | IC50 | 2 | — | |
KARVIVULTZYCNP
|
6.2 | IC50 | 2 | — | |
NPQKNKYIENOLIA
|
6.2 | IC50 | 2 | — | |
ZELZMZDZQZKANU
|
6.2 | IC50 | 2 | — | |
YGXPAGSHLFJKFV
|
6.1 | Ki | 2 | — | |
UVRGHEYADYBWFL
|
6.1 | IC50 | 2 | — | |
SFLFAQAYQIAVDW
|
6.1 | IC50 | 2 | — |