Target Details
| UniProt AC | Q92633 |
|---|---|
| Gene Symbol | LPAR1 |
| Protein Name | Lysophosphatidic acid receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 122
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (8)
Active Molecules (122)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEBSTCAWUQVIOV
|
7.5 | IC50 | 2 | — | |
SVNWCVFZMPJBLW
|
7.5 | IC50 | 2 | — | |
UBQWZKKHKXFYKG
|
7.5 | IC50 | 2 | — | |
SOSAKGSLKXKLFU
|
7.5 | IC50 | 2 | — | |
WFNXESYFHAMZSY
|
7.5 | Ki | 2 | — | |
YOVTYVMJDJNYKX
|
7.5 | IC50 | 2 | — | |
IEJGGFJTLXGJPD
|
7.5 | IC50 | 2 | — | |
SWATWOUWJLKSFA
|
7.5 | IC50 | 2 | — | |
GUCWMYPGSTXNQO
|
7.4 | IC50 | 2 | — | |
LKYKLVDCGBTNJZ
|
7.4 | IC50 | 2 | — | |
ADACZCWUHYGVAD
|
7.4 | IC50 | 2 | — | |
SPTAXSFFLMLIAF
|
7.4 | IC50 | 2 | — | |
WKODFGZRSIFURU
|
7.4 | IC50 | 2 | — | |
IXNPTKKSRPZDOX
|
7.4 | IC50 | 2 | — | |
DYBZGLVYMXXJHF
|
7.4 | IC50 | 2 | — | |
HKSCEHNRNXWQAZ
|
7.3 | IC50 | 2 | — | |
LEZVXIZCJXKBJY
|
7.3 | IC50 | 2 | — | |
LJVDDAKSLFFVPC
|
7.3 | IC50 | 2 | — | |
XGFDCDKWZWQHSI
|
7.3 | IC50 | 2 | — | |
ZZDYCPYBHLLDPA
|
7.3 | IC50 | 2 | — | |
AMBBSDZKBNQSJQ
|
7.3 | IC50 | 2 | — | |
CMQWTHVXHRXUNC
|
7.3 | IC50 | 2 | — | |
GDOYFVLMJDQTQW
|
7.3 | IC50 | 2 | — | |
PZASAAIJIFDWSB
|
7.3 | IC50 | 2 | — | |
FPIPBUXXFQRFKI
|
7.2 | IC50 | 2 | — | |
ISKOLAMFIRHJSH
|
7.2 | IC50 | 2 | — | |
OZBNMNTVTKQCSS
|
7.2 | IC50 | 2 | — | |
HRBIOAKICQOPBD
|
7.2 | IC50 | 2 | — | |
HVANCKKENVXQOH
|
7.2 | IC50 | 2 | — | |
CSFMYMIHKKPMPF
|
7.2 | IC50 | 2 | — | |
HFYPTENHTPNXGP
|
7.2 | IC50 | 3 | — | |
XWQJXYFTQBSZFA
|
7.1 | IC50 | 2 | — | |
FFMZNYWFUDQTJJ
|
7.1 | Ki | 2 | — | |
IGYITFLQCJEIPG
|
7.1 | IC50 | 2 | — | |
QGFGIQUXZJXHPN
|
7.0 | IC50 | 2 | — | |
ZLXAJSGLSQMZJQ
|
7.0 | IC50 | 2 | — | |
GGHASMDNUJBHLO
|
7.0 | IC50 | 2 | — | |
LJTQGSYFZPTOOH
|
7.0 | IC50 | 2 | — | |
XHZMTTZICDAOHN
|
7.0 | IC50 | 2 | — | |
FPBSEOINXWDZPK
|
6.9 | IC50 | 2 | — | |
HXSHFJUOZDIYAO
|
6.9 | IC50 | 2 | — | |
BIVGLZVHXLZIGP
|
6.9 | IC50 | 2 | — | |
PHXJFMYKLBONBN
|
6.8 | Ki | 2 | — | |
ONHLWLKFAFELOK
|
6.8 | IC50 | 2 | — | |
HLVKVWDSLLFMSX
|
6.8 | Ki | 4 | — | |
JGCATLCTRCCGRP
|
6.8 | Ki | 4 | — | |
SGNXTFIPFVFVIJ
|
6.8 | IC50 | 2 | — | |
WBAUSFZQQFMBCS
|
6.8 | IC50 | 2 | — | |
WSECLOSWBXLDEI
|
6.7 | IC50 | 2 | — | |
PLCCQSPJUXGEHV
|
6.7 | IC50 | 2 | — |