Target Details
| UniProt AC | Q92633 |
|---|---|
| Gene Symbol | LPAR1 |
| Protein Name | Lysophosphatidic acid receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 122
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (8)
Active Molecules (122)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WPZAXTRVIVQZCI
|
9.5 | IC50 | 2 | — | |
UQNKBZRQZWHMCX
|
9.4 | IC50 | 2 | — | |
FDOHMOXGKUEJTN
|
9.0 | IC50 | 2 | — | |
YRJOPHXVYGKSJE
|
9.0 | IC50 | 2 | — | |
JAYQKBXYZDGMIP
|
8.7 | IC50 | 2 | — | |
SVXWWGNELSAEBU
|
8.7 | IC50 | 2 | — | |
TUJRAPFNMIKFSP
|
8.6 | IC50 | 2 | — | |
XXIOBZYOOQRDDS
|
8.5 | IC50 | 2 | — | |
DAOODVJVNUBOQM
|
8.5 | IC50 | 2 | — | |
BETITZCZDCWBIT
|
8.4 | IC50 | 2 | — | |
DCOUVLUIDXWAHJ
|
8.4 | IC50 | 2 | — | |
UCZBTVNWIVAWQV
|
8.4 | IC50 | 2 | — | |
HDFMOQYPAALHKY
|
8.3 | IC50 | 2 | — | |
QJPALRLVHVLFGD
|
8.3 | IC50 | 2 | — | |
WRGQSWVCFNIUNZ
|
8.2 | Kd | 3 | — | |
SBSMAUZISCRYBE
|
8.2 | IC50 | 2 | — | |
UIJGNVZGTKKTFL
|
8.2 | IC50 | 2 | — | |
GVJMWLZACNDRBC
|
8.2 | IC50 | 2 | — | |
HWJQFBVAJFHIFS
|
8.2 | IC50 | 2 | — | |
KBJKDHCJCODDDD
|
8.2 | IC50 | 2 | — | |
QSIZRACEBIMNLS
|
8.2 | IC50 | 2 | — | |
YWQLQJKICKYUSN
|
8.2 | IC50 | 2 | — | |
NJJLCPDOBBYPTD
|
8.1 | IC50 | 2 | — | |
PWSIYWWRGAIYIF
|
8.1 | IC50 | 2 | — | |
BKRGCMOFALKWJU
|
8.0 | IC50 | 2 | — | |
QUAWJVQPHQSFAD
|
8.0 | IC50 | 2 | — | |
SRMPREPTJSSCOQ
|
8.0 | IC50 | 2 | — | |
URJZKDCTMMXNDL
|
8.0 | IC50 | 2 | — | |
FPSBJDJNQIVNIK
|
7.9 | IC50 | 2 | — | |
AXNASFMPKJGIGO
|
7.9 | IC50 | 2 | — | |
HWJQFBVAJFHIFS
|
7.9 | IC50 | 2 | — | |
OSXBWRMTMQOKLS
|
7.9 | IC50 | 2 | — | |
RZBDSWRRWUATTL
|
7.9 | IC50 | 2 | — | |
FRPHXCIHOZPOPE
|
7.8 | IC50 | 2 | — | |
ZGDVUUZJQBVBNQ
|
7.8 | IC50 | 2 | — | |
HNCSBMWLHBTZMT
|
7.8 | IC50 | 2 | — | |
UBQWZKKHKXFYKG
|
7.8 | IC50 | 2 | — | |
KYUUSQMQCHIHII
|
7.8 | IC50 | 2 | — | |
HKSCEHNRNXWQAZ
|
7.7 | IC50 | 2 | — | |
AFZOCQFROPJVCM
|
7.7 | IC50 | 2 | — | |
VTJPSPQBNJNSKO
|
7.7 | IC50 | 2 | — | |
ZNPWHDPODRSYQC
|
7.7 | IC50 | 2 | — | |
XTKOCFGCADABCN
|
7.7 | IC50 | 2 | — | |
IKJZZCLSUSZHFO
|
7.6 | IC50 | 2 | — | |
JVVMHUKOPHTRQV
|
7.6 | IC50 | 2 | — | |
MUHRSYPHUZBZJQ
|
7.6 | IC50 | 2 | — | |
YDPWARFVVQLMEY
|
7.6 | IC50 | 2 | — | |
BJSOAPDSLUIFGK
|
7.6 | IC50 | 2 | — | |
NUMUOXFQLCJLCA
|
7.5 | IC50 | 2 | — | |
ZKTDXQOVMQAYEG
|
7.5 | IC50 | 2 | — |