Target Details
| UniProt AC | Q92630 |
|---|---|
| Gene Symbol | DYRK2 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 336
- Clinical molecules 6
- Avg pChEMBL 6.81
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OQSBQXVIMQMCES
|
6.2 | IC50 | 9 | — | |
YGVLUDLFNRZMNT
|
6.2 | IC50 | 8 | — | |
KOMXYYABYRRJBD
|
6.1 | IC50 | 3 | — | |
QVLJVHWQAKYGQI
|
6.1 | IC50 | 8 | — | |
WSUWIXYPBRLNOT
|
6.1 | IC50 | 4 | — | |
LGCHSPYDLIKTIC
|
6.1 | IC50 | 6 | — | |
NZVIEGVPMXNSJT
|
6.1 | IC50 | 2 | — | |
IRBWROIEALHOPH
|
6.1 | IC50 | 7 | — | |
ZYVXTMKTGDARKR
|
6.1 | IC50 | 6 | — | |
BHDRCBRVTBITOC
|
6.1 | IC50 | 2 | — | |
XQQYRDDJENLAME
|
6.1 | IC50 | 8 | — | |
XTJRKTBELWGSDN
|
6.1 | IC50 | 8 | — | |
YSBCFQVEEKUZSU
|
6.1 | IC50 | 9 | — | |
KCTCLVINURCCIL
|
6.1 | IC50 | 7 | — | |
UBUJLBVNZCRWPX
|
6.1 | IC50 | 7 | — | |
BKIAHCJPMJSHSQ
|
6.1 | IC50 | 6 | — | |
CWGKHYILSMYODL
|
6.1 | IC50 | 2 | — | |
HHSNDNONCUTNQR
|
6.1 | IC50 | 7 | — | |
UKFPGYWBGLNLOJ
|
6.1 | IC50 | 2 | — | |
WLUFZZMAAGDSJH
|
6.1 | IC50 | 4 | — | |
WFOMWAYINPJPDX
|
6.1 | IC50 | 9 | — | |
AYTIPFHOSNFHGV
|
6.1 | IC50 | 5 | — | |
DPSFKKBIIZTWDA
|
6.1 | IC50 | 3 | — | |
VGWCJGBQHCMHNJ
|
6.1 | IC50 | 8 | — | |
BXNJHAXVSOCGBA
|
6.0 | IC50 | 14 | — | |
HAFFBDGNUZMNIJ
|
6.0 | IC50 | 7 | — | |
CBTNARFZVOPLBO
|
6.0 | IC50 | 5 | — | |
OEVQTWCGWDOIFZ
|
6.0 | IC50 | 7 | — | |
CTXSEYUOXKGIMM
|
6.0 | IC50 | 3 | — | |
DSQFWMPIQBMOJL
|
6.0 | IC50 | 5 | — | |
MYKOWOGZBMOVBJ
|
6.0 | IC50 | 9 | — | |
BLMDVYRPCVHXPK
|
6.0 | IC50 | 6 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
UZLHPXPKYRQXJV
|
6.0 | IC50 | 2 | — |