Target Details
| UniProt AC | Q92630 |
|---|---|
| Gene Symbol | DYRK2 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 336
- Clinical molecules 6
- Avg pChEMBL 6.81
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YDTHCIZMSQZYMR
|
6.3 | IC50 | 9 | — | |
FABGVXWXZKTQBP
|
6.3 | IC50 | 2 | — | |
JJUHKRNDDMOYGK
|
6.3 | IC50 | 3 | — | |
PMDAVRLCSZSLRH
|
6.3 | Kd | 13 | — | |
PKEDBIGNILOTHW
|
6.3 | IC50 | 3 | — | |
DXVSNYWBRDTHFF
|
6.3 | IC50 | 7 | — | |
SZOYOCHRMSEEMG
|
6.3 | IC50 | 7 | — | |
BNEMOONNXBNRSX
|
6.3 | IC50 | 2 | — | |
OZGASTZOHHWYOH
|
6.3 | IC50 | 3 | — | |
OZGASTZOHHWYOH
|
6.3 | IC50 | 2 | — | |
RUQXGVGYNKIGJD
|
6.3 | IC50 | 7 | — | |
SJWUVVGOTOMGOH
|
6.3 | IC50 | 9 | — | |
USYASDQVUTWEQM
|
6.3 | IC50 | 9 | — | |
BWKADHBOXYDZFU
|
6.3 | IC50 | 10 | — | |
MCNDTHVVURYHKT
|
6.3 | IC50 | 8 | — | |
QCLXNOBXQUWUEW
|
6.3 | IC50 | 9 | — | |
PVFNDFZQGWYILU
|
6.3 | IC50 | 3 | — | |
URXJBXVGNBGIJA
|
6.3 | IC50 | 9 | — | |
BIQADQASLLQRRS
|
6.3 | IC50 | 2 | — | |
FBURYRMHEHTVED
|
6.3 | IC50 | 9 | — | |
ATXGVVQAUKKFAN
|
6.2 | IC50 | 4 | — | |
DXVSNYWBRDTHFF
|
6.2 | IC50 | 10 | — | |
NPQSOFKMVBBVFF
|
6.2 | IC50 | 2 | — | |
OYDWEMSWMQKSLK
|
6.2 | IC50 | 8 | — | |
RAQBQAXSLHDSKW
|
6.2 | IC50 | 8 | — | |
ANKYADWZYKSCAJ
|
6.2 | IC50 | 7 | — | |
GEJSQZULGDKBQV
|
6.2 | IC50 | 8 | — | |
LOLPPWBBNUVNQZ
|
6.2 | IC50 | 97 | Yes | |
RLTCEYSNDOXWKS
|
6.2 | IC50 | 7 | — | |
UDBMFFIMVBBFKP
|
6.2 | IC50 | 3 | — | |
YKFHBMIPXGSMRS
|
6.2 | IC50 | 7 | — | |
QVYXLOYBJBMXNP
|
6.2 | IC50 | 7 | — | |
OJYINLHOEHUFHI
|
6.2 | IC50 | 7 | — | |
PDJLHUHTIYCYTA
|
6.2 | IC50 | 4 | — | |
KQZBWTMAFLOSPA
|
6.2 | IC50 | 8 | — | |
MVRRAWJPZXNFMK
|
6.2 | IC50 | 6 | — | |
QCHDHJOEPUQALZ
|
6.2 | IC50 | 9 | — | |
YMIDGKZVYFXIBW
|
6.2 | IC50 | 8 | — | |
DXVSNYWBRDTHFF
|
6.2 | IC50 | 9 | — | |
GPMRASYSIQENIJ
|
6.2 | IC50 | 3 | — | |
JYRRTOFZIGEMAN
|
6.2 | IC50 | 2 | — | |
BEILWJKGWBDPRG
|
6.2 | IC50 | 7 | — | |
CBTNARFZVOPLBO
|
6.2 | IC50 | 8 | — | |
ZBKFRVXDYILXFJ
|
6.2 | IC50 | 6 | — | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
AUSDRYPYNGBOOX
|
6.2 | IC50 | 2 | — | |
XCTYEZWILVGTGO
|
6.2 | IC50 | 9 | — | |
AHHFGEKSWVBFGA
|
6.2 | IC50 | 3 | — | |
AHHFGEKSWVBFGA
|
6.2 | IC50 | 2 | — | |
CHQYAWLKOUOTQO
|
6.2 | IC50 | 7 | — |