Target Details
| UniProt AC | Q92630 |
|---|---|
| Gene Symbol | DYRK2 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 336
- Clinical molecules 6
- Avg pChEMBL 6.81
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SOHWYEVCBPDAIO
|
6.5 | IC50 | 3 | — | |
HTNKXRHQVGPWRO
|
6.5 | IC50 | 3 | — | |
NAYXGFSGXGZZCZ
|
6.5 | IC50 | 3 | — | |
DCHAEDURAZJASA
|
6.5 | IC50 | 9 | — | |
UXIAMCZUNQBRTJ
|
6.5 | IC50 | 4 | — | |
NZMFVJNZGKELJC
|
6.5 | IC50 | 4 | — | |
OBKVROGZKBOQSW
|
6.5 | IC50 | 3 | — | |
OBKVROGZKBOQSW
|
6.5 | IC50 | 2 | — | |
XTJRKTBELWGSDN
|
6.5 | IC50 | 8 | — | |
CVIZQDCZKWMREN
|
6.5 | IC50 | 2 | — | |
UCJUQIKMOSVOJR
|
6.5 | IC50 | 2 | — | |
LMXLOYKFDZEHCS
|
6.5 | IC50 | 7 | — | |
ROPFCXUWNMYMSW
|
6.5 | IC50 | 10 | — | |
FANUXQYVRUHAAH
|
6.4 | IC50 | 6 | — | |
IFLBFWBMAWIBBZ
|
6.4 | Kd | 7 | — | |
HMMICWRUNSZYCJ
|
6.4 | IC50 | 3 | — | |
JBWDTSLHUJHODF
|
6.4 | IC50 | 9 | — | |
SZOYOCHRMSEEMG
|
6.4 | IC50 | 3 | — | |
BULHRWBHKAVJMT
|
6.4 | IC50 | 8 | — | |
FTGAOPZDJRWUTG
|
6.4 | IC50 | 6 | — | |
OVVHFDIQCYTOAS
|
6.4 | IC50 | 9 | — | |
SJYQOVMGZOATNK
|
6.4 | IC50 | 9 | — | |
WFOMWAYINPJPDX
|
6.4 | IC50 | 9 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
CIJWGWNHXQYIJC
|
6.4 | IC50 | 5 | — | |
FJAIARRQBXWUMX
|
6.4 | IC50 | 2 | — | |
IDOKKOQIQLHASZ
|
6.4 | IC50 | 8 | — | |
JBWDTSLHUJHODF
|
6.4 | IC50 | 8 | — | |
MLAPBLMPGXKRBF
|
6.4 | IC50 | 3 | — | |
SKKBUBMBPCJYKW
|
6.4 | IC50 | 9 | — | |
DHUALHRRYFDDKC
|
6.4 | IC50 | 2 | — | |
XVVPNHZWUXCHJE
|
6.4 | IC50 | 3 | — | |
ANKYADWZYKSCAJ
|
6.4 | IC50 | 7 | — | |
IJFKKIMDRSZOOW
|
6.4 | IC50 | 6 | — | |
QZIYOWZOZNSBGJ
|
6.4 | IC50 | 3 | — | |
UMWJBFSPIYCGRG
|
6.4 | IC50 | 7 | — | |
WREJZZXSNOJGIW
|
6.4 | IC50 | 8 | — | |
HJEKFRDOAYXXRU
|
6.4 | IC50 | 8 | — | |
PKEDBIGNILOTHW
|
6.4 | IC50 | 2 | — | |
PKEDBIGNILOTHW
|
6.4 | IC50 | 5 | — | |
WBCONKPHYUGGFA
|
6.4 | IC50 | 3 | — | |
CYVGSDYVNUNREA
|
6.4 | IC50 | 5 | — | |
FIVWKNZKXNNFCW
|
6.4 | IC50 | 9 | — | |
GVANUSPDJMCBIK
|
6.4 | IC50 | 6 | — | |
XNYOTZHBHJIMBV
|
6.4 | IC50 | 2 | — | |
YKDZIFFKQUNVHH
|
6.4 | IC50 | 3 | — | |
JBWDTSLHUJHODF
|
6.3 | IC50 | 9 | — | |
NNPWUWSWEGWPMQ
|
6.3 | IC50 | 8 | — | |
IJFKKIMDRSZOOW
|
6.3 | IC50 | 8 | — | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — |