Target Details
| UniProt AC | Q92630 |
|---|---|
| Gene Symbol | DYRK2 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 336
- Clinical molecules 6
- Avg pChEMBL 6.81
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OWDVXJJCVWTPPW
|
6.8 | IC50 | 8 | — | |
WHPORTUXBLFUPA
|
6.8 | IC50 | 9 | — | |
SBYPANVVFZBWDF
|
6.8 | IC50 | 9 | — | |
AMUFSGPBIFOSNV
|
6.7 | IC50 | 3 | — | |
KBMQGIPVJGXLOU
|
6.7 | IC50 | 7 | — | |
LXQXBEIFOYAXOP
|
6.7 | IC50 | 9 | — | |
OQGLPYHETIJRBX
|
6.7 | IC50 | 3 | — | |
OQGLPYHETIJRBX
|
6.7 | IC50 | 3 | — | |
VBYRFFCBZNEHAL
|
6.7 | IC50 | 4 | — | |
HIDZIHZHRJJHIB
|
6.7 | IC50 | 2 | — | |
POSGRZQCKOTBHE
|
6.7 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.7 | IC50 | 408 | — | |
CHQYAWLKOUOTQO
|
6.7 | IC50 | 20 | — | |
CIICGXXZCWRFQE
|
6.7 | IC50 | 7 | — | |
CQZSVQKINMHLBO
|
6.7 | IC50 | 4 | — | |
FWFWXUJORMCFKY
|
6.7 | IC50 | 3 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
OGPJOAYIAOEJAM
|
6.7 | IC50 | 8 | — | |
WQYUNADCLFWKGN
|
6.7 | IC50 | 7 | — | |
LAMQDGYKYXRPLW
|
6.7 | IC50 | 2 | — | |
MEKFXUFACKZUCV
|
6.7 | IC50 | 9 | — | |
PVKHDYBJGIJIAB
|
6.7 | IC50 | 2 | — | |
WGBRJADREQKUMW
|
6.7 | IC50 | 2 | — | |
XSEOLUNNBOQVET
|
6.7 | IC50 | 3 | — | |
GCSZJMUFYOAHFY
|
6.7 | IC50 | 8 | — | |
ACOQCSBMVFAWQV
|
6.6 | IC50 | 8 | — | |
SGWXBOBKZVIVOW
|
6.6 | IC50 | 3 | — | |
SGWXBOBKZVIVOW
|
6.6 | IC50 | 3 | — | |
YRFAWSIUIFNVQA
|
6.6 | IC50 | 9 | — | |
BXPPINFBXDOAPI
|
6.6 | IC50 | 2 | — | |
GHQYHWMWJLSKRP
|
6.6 | IC50 | 9 | — | |
LVSVYVPFNYRNOF
|
6.6 | IC50 | 8 | — | |
RUQXGVGYNKIGJD
|
6.6 | IC50 | 9 | — | |
BBCSUMURJUYILA
|
6.6 | IC50 | 9 | — | |
QGGNWMQODZFHNG
|
6.6 | IC50 | 4 | — | |
HGMCNIGKEVZHFM
|
6.6 | IC50 | 8 | — | |
RLTCEYSNDOXWKS
|
6.6 | IC50 | 9 | — | |
RYWACTNAXCMTTN
|
6.6 | IC50 | 9 | — | |
WHPORTUXBLFUPA
|
6.6 | IC50 | 8 | — | |
DJHMDVUOYUYLOJ
|
6.6 | IC50 | 9 | — | |
FIVWKNZKXNNFCW
|
6.6 | IC50 | 8 | — | |
MCHFBGTXGSLCLO
|
6.6 | IC50 | 2 | — | |
YJKPCYDSZXIODK
|
6.6 | IC50 | 8 | — | |
YORVMWUGDVGXOQ
|
6.6 | IC50 | 8 | — | |
BBCSUMURJUYILA
|
6.5 | IC50 | 10 | — | |
ONCJKEZPQVEATH
|
6.5 | IC50 | 2 | — | |
JFDRONLMXPRQPP
|
6.5 | IC50 | 9 | — | |
QTRZNDLLYHSJSH
|
6.5 | IC50 | 9 | — | |
AVLYNJZZQYEFEA
|
6.5 | IC50 | 8 | Yes | |
RCYPVQCPYKNSTG
|
6.5 | IC50 | 7 | — |