Target Details
| UniProt AC | Q92630 |
|---|---|
| Gene Symbol | DYRK2 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 336
- Clinical molecules 6
- Avg pChEMBL 6.81
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJWUVVGOTOMGOH
|
7.0 | IC50 | 12 | — | |
SLKHMZQUNIHINK
|
7.0 | IC50 | 10 | — | |
MUOKSQABCJCOPU
|
7.0 | IC50 | 36 | — | |
SQWZFLMPDUSYGV
|
7.0 | IC50 | 11 | — | |
SQWZFLMPDUSYGV
|
7.0 | IC50 | 8 | — | |
UGUVGLVHRPLWRS
|
7.0 | IC50 | 3 | — | |
UGUVGLVHRPLWRS
|
7.0 | IC50 | 3 | — | |
OVRDWLJZSQZCBW
|
7.0 | IC50 | 2 | — | |
AINKQRBPBUTJRM
|
7.0 | IC50 | 5 | — | |
DYIOAOFYWZXKEX
|
7.0 | IC50 | 4 | — | |
DYIOAOFYWZXKEX
|
7.0 | IC50 | 4 | — | |
IJFKKIMDRSZOOW
|
7.0 | IC50 | 9 | — | |
JXQZHHAAJMQJKU
|
7.0 | IC50 | 9 | — | |
SJWUVVGOTOMGOH
|
7.0 | IC50 | 10 | — | |
YHZQZEGQCKWCLP
|
7.0 | IC50 | 9 | — | |
CCUMIOKJQCVBML
|
6.9 | IC50 | 2 | — | |
CCUMIOKJQCVBML
|
6.9 | IC50 | 2 | — | |
QTHCAAFKVUWAFI
|
6.9 | IC50 | 23 | — | |
JDNVNTCGESXSFD
|
6.9 | IC50 | 4 | — | |
LZRHAZRGHSSHLR
|
6.9 | IC50 | 7 | — | |
PRJNNPMIUGYOST
|
6.9 | IC50 | 14 | — | |
YELPLVUUDHOICI
|
6.9 | IC50 | 4 | — | |
YSODDCRKIDDXKM
|
6.9 | IC50 | 9 | — | |
IVSYLIPATGYBCZ
|
6.9 | IC50 | 7 | — | |
DOWFKLSBHHHHTF
|
6.9 | IC50 | 4 | — | |
WYQPGNJIFZHADC
|
6.9 | IC50 | 2 | — | |
ZBYBDKHFLSHGBP
|
6.9 | IC50 | 4 | — | |
ZBYBDKHFLSHGBP
|
6.9 | IC50 | 4 | — | |
IQPGVUQARGVQGU
|
6.9 | IC50 | 2 | — | |
QTRZNDLLYHSJSH
|
6.9 | IC50 | 9 | — | |
XKBACCJVCIHQMK
|
6.9 | IC50 | 2 | — | |
VCCCOYOXNKTQFO
|
6.9 | IC50 | 9 | — | |
KYOPCGIPHGGWMV
|
6.8 | IC50 | 7 | — | |
BDMXFIMYKGLQAL
|
6.8 | IC50 | 9 | — | |
UGYUFJPHSWYELP
|
6.8 | IC50 | 8 | — | |
ZXNKLLQATJHCGU
|
6.8 | IC50 | 2 | — | |
YAXGFAAKCUOWNM
|
6.8 | IC50 | 9 | — | |
LZUJDIWVWSRLRQ
|
6.8 | IC50 | 4 | — | |
LZUJDIWVWSRLRQ
|
6.8 | IC50 | 4 | — | |
PEXTWZUAIQCVBB
|
6.8 | IC50 | 3 | — | |
YORVMWUGDVGXOQ
|
6.8 | IC50 | 8 | — | |
AMBKAVGTUWUVBS
|
6.8 | IC50 | 8 | — | |
YHZQZEGQCKWCLP
|
6.8 | IC50 | 9 | — | |
UUIPRATXTHJYHH
|
6.8 | IC50 | 3 | — | |
ZHTZVZJNJGCSJO
|
6.8 | IC50 | 7 | — | |
MQRHLOPPMRFMKM
|
6.8 | IC50 | 9 | — | |
USSKXRGFNVFHFF
|
6.8 | IC50 | 7 | — | |
UTDNMHFLZJFPPY
|
6.8 | IC50 | 4 | — | |
MIEPXFZAJZPNFG
|
6.8 | IC50 | 5 | — | |
MIEPXFZAJZPNFG
|
6.8 | IC50 | 8 | — |