Target Details
| UniProt AC | Q92630 |
|---|---|
| Gene Symbol | DYRK2 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 336
- Clinical molecules 6
- Avg pChEMBL 6.81
Active Molecules (336)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKCITBQBYLZFBK
|
7.5 | IC50 | 3 | — | |
QCTMVDQWYGRUJK
|
7.5 | IC50 | 9 | — | |
UUXDJIVNVOOKFQ
|
7.5 | IC50 | 9 | — | |
WXMYTQDKBPDSSR
|
7.5 | IC50 | 4 | — | |
QXPJTIYARGTANC
|
7.5 | IC50 | 3 | — | |
GTVWYIASBVPCEA
|
7.5 | IC50 | 2 | — | |
PGPHHJBZEGSUNE
|
7.5 | IC50 | 4 | — | |
SDQPABOSBRYYPV
|
7.5 | IC50 | 2 | — | |
ZQZULRTVXPNQNP
|
7.5 | IC50 | 4 | — | |
GXCOUFPTCZUTEE
|
7.4 | IC50 | 10 | — | |
JANQPHRPUAYQTA
|
7.4 | IC50 | 5 | — | |
QULVCQWDONFUCP
|
7.4 | IC50 | 2 | — | |
ABRIIMZXUFHPCH
|
7.4 | IC50 | 5 | — | |
HEVBCYZPXGZFGS
|
7.4 | IC50 | 11 | — | |
WEQRXDXDFLBIDK
|
7.4 | IC50 | 8 | — | |
WNKQZLFWZLQFOH
|
7.4 | IC50 | 3 | — | |
PBGPFWACZLCJFH
|
7.4 | IC50 | 3 | — | |
RGKOSKZCLZXDJI
|
7.4 | IC50 | 4 | — | |
YGXHQYJKJUFSJI
|
7.4 | IC50 | 14 | — | |
ITOTZLBIDAOTGK
|
7.3 | IC50 | 4 | — | |
ITOTZLBIDAOTGK
|
7.3 | IC50 | 4 | — | |
PUGXENIKUPHCAF
|
7.3 | IC50 | 3 | — | |
DSCUTYQYWCTFQL
|
7.3 | IC50 | 6 | — | |
KAGWQDFFFLWBFD
|
7.3 | IC50 | 8 | — | |
YEZMGVBTPDYRPO
|
7.3 | IC50 | 8 | — | |
IOUKAQLHORTKRT
|
7.3 | IC50 | 3 | — | |
MWQLICNQHCLBLQ
|
7.3 | IC50 | 3 | — | |
CGPYAXSYKQBYKJ
|
7.2 | IC50 | 12 | — | |
MFAQYJIYDMLAIM
|
7.2 | Kd | 130 | Yes | |
FMOOGIYSVBVFIT
|
7.2 | IC50 | 2 | — | |
BUDHVVXPBGMAPV
|
7.2 | IC50 | 11 | — | |
BWNQBFHVFFZHMR
|
7.2 | IC50 | 10 | — | |
FGBSSPMQGRUJPS
|
7.2 | IC50 | 10 | — | |
QMUKOEKTUBVPFU
|
7.2 | IC50 | 12 | — | |
UZWDCWONPYILKI
|
7.2 | IC50 | 47 | — | |
BPNUQXPIQBZCMR
|
7.2 | Kd | 83 | Yes | |
MOYYMSNZEWQWQJ
|
7.2 | IC50 | 3 | — | |
OHARPIGKJAKOCM
|
7.2 | IC50 | 8 | — | |
PGPHHJBZEGSUNE
|
7.1 | IC50 | 21 | — | |
PGPHHJBZEGSUNE
|
7.1 | IC50 | 17 | — | |
OAKDCYWBXLUPQD
|
7.1 | IC50 | 4 | — | |
QXFBTYPBHYOEMX
|
7.1 | IC50 | 9 | — | |
HFLXYSRIPKXGOQ
|
7.1 | IC50 | 4 | — | |
VCFPJHJKTXRDGD
|
7.1 | IC50 | 3 | — | |
RVNDFXJEYCICIV
|
7.1 | IC50 | 7 | — | |
QKGQVNUHCXZGQO
|
7.1 | IC50 | 2 | — | |
RRJNXBNVQSVJBA
|
7.1 | IC50 | 2 | — | |
NBTJWRPKGNQBJS
|
7.0 | IC50 | 8 | — | |
DCJOTKUJWJFCSP
|
7.0 | IC50 | 9 | — | |
DYHKEGKDOOZETF
|
7.0 | IC50 | 9 | — |