Target Details
| UniProt AC | Q8WYR1 |
|---|---|
| Gene Symbol | PIK3R5 |
| Protein Name | Phosphoinositide 3-kinase regulatory subunit 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10486 (PI3K_1B_p101) |
Summary
- Multi-target molecules 297
- Clinical molecules 1
- Avg pChEMBL 6.75
KEGG Pathways (11)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Kaposi sarcoma-associated herpesvirus infection
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (297)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHYGZQVJMLTYPP
|
6.2 | IC50 | 8 | — | |
NQGQCKYICODPRT
|
6.2 | IC50 | 8 | — | |
SWHDQTHOFGUWTP
|
6.2 | IC50 | 8 | — | |
WKHVREDXOZYDKG
|
6.2 | IC50 | 8 | — | |
YGYMLYFXPLWCSP
|
6.2 | IC50 | 8 | — | |
AHWHGALWRKOGIW
|
6.2 | IC50 | 8 | — | |
JBEDJEOXQRSVHA
|
6.2 | IC50 | 8 | — | |
PGOGWPYCIZVYBQ
|
6.2 | IC50 | 8 | — | |
PUOJAIRQIFIHLD
|
6.2 | IC50 | 8 | — | |
AJNVYCYEQWOCQG
|
6.2 | IC50 | 8 | — | |
PRANHWURGNZBDG
|
6.2 | IC50 | 8 | — | |
ALNSNMBSENGUSM
|
6.1 | IC50 | 8 | — | |
OBWJIWMQAUQEMB
|
6.1 | IC50 | 8 | — | |
VWNUIZMUGGBKPQ
|
6.1 | IC50 | 8 | — | |
WXQSAROWLFBICE
|
6.1 | IC50 | 8 | — | |
XFROLARWNLOEQS
|
6.1 | IC50 | 8 | — | |
LAXCPCHPIFTFEJ
|
6.1 | IC50 | 8 | — | |
RJPQDGBWPPNUQX
|
6.1 | IC50 | 8 | — | |
KANIKZLNGVDVBI
|
6.1 | IC50 | 8 | — | |
MBCLTTATBWHRGR
|
6.1 | IC50 | 8 | — | |
WJCYHWGNDVBBPJ
|
6.1 | IC50 | 8 | — | |
LLSPYQXCBDPCKL
|
6.1 | IC50 | 8 | — | |
MIFBYDPTRPDGOS
|
6.1 | IC50 | 8 | — | |
GWZVMSSDIBHICV
|
6.1 | IC50 | 8 | — | |
HTFVOKCSBZNVCM
|
6.1 | IC50 | 8 | — | |
NORWTLLCOTYPQA
|
6.1 | IC50 | 8 | — | |
NUVNLRITBKISJS
|
6.1 | IC50 | 8 | — | |
UKYZNGMYDHPKCT
|
6.1 | IC50 | 8 | — | |
MEDJQGQNXIYESM
|
6.1 | IC50 | 8 | — | |
XQTHYNKOCLMRDN
|
6.1 | IC50 | 8 | — | |
ZQMRWZWYYAEHCM
|
6.1 | IC50 | 8 | — | |
NNJFATAWXWTKJW
|
6.0 | IC50 | 8 | — | |
XMIXKIYGSBKJHW
|
6.0 | IC50 | 8 | — | |
BZTIAAOQYKUYMP
|
6.0 | IC50 | 8 | — | |
CDCYZIADQZZXOR
|
6.0 | IC50 | 8 | — | |
DLBMZAAMUILROS
|
6.0 | IC50 | 8 | — | |
DPXYTFRWYCEDNN
|
6.0 | IC50 | 8 | — | |
GRNHQFWGZJVSRA
|
6.0 | IC50 | 8 | — | |
NLTSUUCKGVRGEB
|
6.0 | IC50 | 8 | — | |
TWYYRCNMQXRTJG
|
6.0 | IC50 | 8 | — | |
XLVLZQZUUOKWBV
|
6.0 | IC50 | 8 | — | |
AGHMOGGRPAZCJV
|
6.0 | IC50 | 8 | — | |
NLPLFNLMHHBEKR
|
6.0 | IC50 | 8 | — | |
RZZKNWAYYKUPNA
|
6.0 | IC50 | 8 | — | |
FJLPTFADSJAOAV
|
6.0 | IC50 | 8 | — | |
LSMFRSSROQIZIC
|
6.0 | IC50 | 8 | — | |
YCDRKRFDMPJHDQ
|
6.0 | IC50 | 8 | — |