Target Details
| UniProt AC | Q8WYR1 |
|---|---|
| Gene Symbol | PIK3R5 |
| Protein Name | Phosphoinositide 3-kinase regulatory subunit 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10486 (PI3K_1B_p101) |
Summary
- Multi-target molecules 297
- Clinical molecules 1
- Avg pChEMBL 6.75
KEGG Pathways (11)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Kaposi sarcoma-associated herpesvirus infection
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (297)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RZNZPAXQLLCDSL
|
6.6 | IC50 | 8 | — | |
XGSGIVHSKLTSTI
|
6.6 | IC50 | 8 | — | |
BMBWVOBMAXRAQV
|
6.6 | IC50 | 8 | — | |
IPJVWNODSCZWCO
|
6.6 | IC50 | 8 | — | |
KXYRGDRFYJGKRS
|
6.6 | IC50 | 8 | — | |
HWQXDWNWVAOPGP
|
6.6 | IC50 | 8 | — | |
QWRWABZPKBNWJW
|
6.6 | IC50 | 8 | — | |
KWRMMGQBGIIMIQ
|
6.6 | IC50 | 8 | — | |
BQQOJYRNJKJNIK
|
6.6 | IC50 | 8 | — | |
YYLPYSXYKVBLBD
|
6.6 | IC50 | 8 | — | |
BSQLGIZDXTZOLY
|
6.5 | IC50 | 8 | — | |
CENMCUFOZLPPKP
|
6.5 | IC50 | 8 | — | |
XGBDKCNPCGGPBO
|
6.5 | IC50 | 8 | — | |
BZQJNLXTYPFQDO
|
6.5 | IC50 | 8 | — | |
HNOFMPKORNQUAT
|
6.5 | IC50 | 8 | — | |
MWFGYPVIIVOLMX
|
6.5 | IC50 | 8 | — | |
ONIZUNGHVJHSTA
|
6.5 | IC50 | 8 | — | |
YYGHWHOJQMMELF
|
6.5 | IC50 | 8 | — | |
DMLMQDOHTGPLQS
|
6.5 | IC50 | 8 | — | |
IOBVXRYCNWSMKS
|
6.5 | IC50 | 8 | — | |
NZBPSKJJETVVOQ
|
6.5 | IC50 | 8 | — | |
DOTAHHROQNVDAF
|
6.5 | IC50 | 8 | — | |
HWBDCKWOZGYXRP
|
6.5 | IC50 | 8 | — | |
LMUCVOYUWPGAFT
|
6.5 | IC50 | 8 | — | |
OBQFGWRYNYWVEO
|
6.5 | IC50 | 8 | — | |
BORRMUVLRFHNSP
|
6.5 | IC50 | 8 | — | |
DJQCYLXTSKHWDY
|
6.5 | IC50 | 8 | — | |
HRJNMMQECAFPDZ
|
6.5 | IC50 | 8 | — | |
JIFVVFLJYNJCGH
|
6.5 | IC50 | 8 | — | |
NFHSJYKXENYICE
|
6.5 | IC50 | 8 | — | |
RWKVSRSWLBMQFZ
|
6.5 | IC50 | 8 | — | |
RGZQZTZWYUCVAY
|
6.5 | IC50 | 8 | — | |
UQOMRZMTEAAICA
|
6.5 | IC50 | 8 | — | |
ZZSPAALVTKNEPM
|
6.5 | IC50 | 8 | — | |
CYJSBMVDFDOPHN
|
6.4 | IC50 | 8 | — | |
DIHKSILZPYDOBE
|
6.4 | IC50 | 8 | — | |
DWTLVZKCLZPGBC
|
6.4 | IC50 | 8 | — | |
HUKWEGRPUKJFER
|
6.4 | IC50 | 8 | — | |
KGTAFFXGCXZNSF
|
6.4 | IC50 | 8 | — | |
MJFBXUGGKSQWGD
|
6.4 | IC50 | 8 | — | |
LMFDSWCIMMUPRR
|
6.4 | IC50 | 8 | — | |
VMLCDXGHZQRAON
|
6.4 | IC50 | 8 | — | |
SPSKNHQNGRNHNA
|
6.4 | IC50 | 8 | — | |
ULDRLGOGVDLJIJ
|
6.4 | IC50 | 8 | — | |
YYDHSDLMQPQAPK
|
6.4 | IC50 | 8 | — | |
ZEETVDFZYSVSGW
|
6.4 | IC50 | 6 | — | |
BSRGPULLSTVXNM
|
6.4 | IC50 | 8 | — | |
SIMPDDFJFTVDMJ
|
6.4 | IC50 | 8 | — | |
ANCWBHOYWBANAV
|
6.4 | IC50 | 8 | — | |
NRULIRPKJVMPDY
|
6.4 | IC50 | 8 | — |