Target Details
| UniProt AC | Q8WYR1 |
|---|---|
| Gene Symbol | PIK3R5 |
| Protein Name | Phosphoinositide 3-kinase regulatory subunit 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10486 (PI3K_1B_p101) |
Summary
- Multi-target molecules 297
- Clinical molecules 1
- Avg pChEMBL 6.75
KEGG Pathways (11)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Kaposi sarcoma-associated herpesvirus infection
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (297)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXSQTDIQFDKYIS
|
6.9 | IC50 | 7 | — | |
LHNIIDJUOCFXAP
|
6.9 | IC50 | 20 | Yes | |
AYRHYIQWAHXGQS
|
6.9 | IC50 | 8 | — | |
MDBPGMMGPFYUIX
|
6.9 | IC50 | 8 | — | |
WTQFUMYRIIWPGE
|
6.9 | IC50 | 8 | — | |
CQOAMUDQCWRECW
|
6.9 | IC50 | 8 | — | |
CWHUFRVAEUJCEF
|
6.9 | IC50 | 8 | — | |
VBARFYIZOQPRIU
|
6.9 | IC50 | 8 | — | |
GLLFQTCFJDJTEY
|
6.9 | IC50 | 8 | — | |
FDEAQYIYQUZQAJ
|
6.9 | IC50 | 8 | — | |
FVCYICGIUXQQRS
|
6.9 | IC50 | 8 | — | |
CRENPEXXTIJKAA
|
6.9 | IC50 | 8 | — | |
VITSWBMXSGIZBK
|
6.8 | IC50 | 8 | — | |
UBWTUXFRFOVNSZ
|
6.8 | IC50 | 8 | — | |
URZITQGEWBAINN
|
6.8 | IC50 | 8 | — | |
DVJHHRDBSCMRFO
|
6.8 | IC50 | 8 | — | |
GCMPYYJJMWUTQX
|
6.8 | IC50 | 8 | — | |
TWSFAEOUABXTKC
|
6.8 | IC50 | 8 | — | |
RCDKXUXYPKPWOL
|
6.8 | IC50 | 8 | — | |
YBSONZDEWIPQTP
|
6.8 | IC50 | 2 | — | |
OQNSHGSWBWLCGD
|
6.8 | IC50 | 8 | — | |
NUBPXPBMWBORQH
|
6.8 | IC50 | 8 | — | |
QINAYZWLPHRNRP
|
6.8 | IC50 | 8 | — | |
XTJYQRUVPWZZMO
|
6.8 | IC50 | 8 | — | |
NFVBVBZCCSWOGV
|
6.8 | IC50 | 8 | — | |
QIIACSBLOYITSG
|
6.8 | IC50 | 8 | — | |
DKBIFPXBCXSLNM
|
6.8 | IC50 | 8 | — | |
DTNRKAREUFEJOT
|
6.8 | IC50 | 8 | — | |
CIEPFNWWFNULHV
|
6.7 | IC50 | 7 | — | |
KXUYUETUZFPOQS
|
6.7 | IC50 | 8 | — | |
OOGFHRAURPOHAA
|
6.7 | IC50 | 8 | — | |
KPFIPJMXDOSFKZ
|
6.7 | IC50 | 8 | — | |
HYFOWZDHZOPTAI
|
6.7 | IC50 | 8 | — | |
MDBPGMMGPFYUIX
|
6.7 | IC50 | 8 | — | |
JXIVPCDJNLIENJ
|
6.7 | IC50 | 8 | — | |
DMLMQDOHTGPLQS
|
6.7 | IC50 | 8 | — | |
SYVHOZRIBZQVSX
|
6.7 | IC50 | 8 | — | |
VUTWTOWSCDWESM
|
6.7 | IC50 | 8 | — | |
SUENWRGZWCPLSE
|
6.7 | IC50 | 8 | — | |
ALTWEBDMLOHYHS
|
6.7 | IC50 | 8 | — | |
ILSRTSOJUBOZBR
|
6.7 | IC50 | 8 | — | |
VPFKGOXBNBHRQI
|
6.7 | IC50 | 8 | — | |
SFNWXIWGLMNMJM
|
6.6 | IC50 | 8 | — | |
XEBPQXAZUWVEBS
|
6.6 | IC50 | 8 | — | |
CZAQUOYKQWEFOR
|
6.6 | IC50 | 8 | — | |
YRFCSVLNUNXFLF
|
6.6 | IC50 | 8 | — | |
IHWJVVJNUJWQEC
|
6.6 | IC50 | 8 | — | |
ILZWGSJNBKEAOZ
|
6.6 | IC50 | 8 | — | |
BHJYMNQXMLXYJW
|
6.6 | IC50 | 8 | — | |
QGXNCNPNSMLJHD
|
6.6 | IC50 | 8 | — |