Target Details
| UniProt AC | Q8WYR1 |
|---|---|
| Gene Symbol | PIK3R5 |
| Protein Name | Phosphoinositide 3-kinase regulatory subunit 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10486 (PI3K_1B_p101) |
Summary
- Multi-target molecules 297
- Clinical molecules 1
- Avg pChEMBL 6.75
KEGG Pathways (11)
- Adrenergic signaling in cardiomyocytes
- Apelin signaling pathway
- Chemokine signaling pathway
- Cholinergic synapse
- Kaposi sarcoma-associated herpesvirus infection
- Oxytocin signaling pathway
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Toxoplasmosis
- cGMP-PKG signaling pathway
Associated Diseases (1)
Active Molecules (297)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PEIFGMMJOLFHBE
|
7.4 | IC50 | 8 | — | |
GIQAVYAYXZICPG
|
7.4 | IC50 | 8 | — | |
YXFHSKVBWDUQIW
|
7.4 | IC50 | 8 | — | |
DZJGDNZVUPCXPX
|
7.4 | IC50 | 8 | — | |
HGAJTKWPNZDTRJ
|
7.3 | IC50 | 8 | — | |
NXHSCEQOULVBJS
|
7.3 | IC50 | 8 | — | |
UDDJJHILDQDTBM
|
7.3 | IC50 | 8 | — | |
AJRVMUXGCPDPOT
|
7.3 | IC50 | 8 | — | |
CQPIITBUFCLJQW
|
7.3 | IC50 | 8 | — | |
KXKADLQRHDFGBR
|
7.3 | IC50 | 8 | — | |
GXTWTBFETNXESR
|
7.3 | IC50 | 8 | — | |
OJCJBVKNUFOBRH
|
7.3 | IC50 | 8 | — | |
KBOCINOJPQBJHY
|
7.3 | IC50 | 8 | — | |
URZITQGEWBAINN
|
7.3 | IC50 | 8 | — | |
DFESDZGEOSBXMQ
|
7.2 | IC50 | 8 | — | |
SUGRZLGNJSNCRI
|
7.2 | IC50 | 8 | — | |
MEDRUYBTHOYYBE
|
7.2 | IC50 | 8 | — | |
MNSRURCAGZOZFY
|
7.2 | IC50 | 8 | — | |
GALWNKLIQPVNFO
|
7.2 | IC50 | 8 | — | |
IVJBBSRYSTWCRD
|
7.2 | IC50 | 8 | — | |
RABFNJUMQFEXTQ
|
7.2 | IC50 | 8 | — | |
UDGRXBYGXYOMBG
|
7.2 | IC50 | 8 | — | |
BXWUMOJSXVZWKL
|
7.1 | IC50 | 8 | — | |
FUMQATBGDGLOKH
|
7.1 | IC50 | 8 | — | |
JJIZJEXAZKGVCY
|
7.1 | IC50 | 8 | — | |
MKPRDFDJZIWWHV
|
7.1 | IC50 | 8 | — | |
VMHQTUFUBQDAPM
|
7.1 | IC50 | 8 | — | |
UDDJJHILDQDTBM
|
7.1 | IC50 | 8 | — | |
HWQXDWNWVAOPGP
|
7.1 | IC50 | 8 | — | |
MUTFYPSFGCHZFO
|
7.1 | IC50 | 2 | — | |
YRTQNKZPRFQKJD
|
7.1 | IC50 | 8 | — | |
YZAOAYLROJTXKO
|
7.1 | IC50 | 8 | — | |
OSLYEXGCLGGXQD
|
7.1 | IC50 | 8 | — | |
RNJXEBWYBBNUDN
|
7.1 | IC50 | 8 | — | |
SNTINYRTBPIKSO
|
7.0 | IC50 | 8 | — | |
ALMGVNBNMXRCQV
|
7.0 | IC50 | 8 | — | |
BQXCOOOANMKMJT
|
7.0 | IC50 | 8 | — | |
GVSPTNBTTDSKBX
|
7.0 | IC50 | 8 | — | |
YYMJOSXPNZYXDU
|
7.0 | IC50 | 8 | — | |
QPTYEYDIOWOEAT
|
7.0 | IC50 | 8 | — | |
GALWNKLIQPVNFO
|
7.0 | IC50 | 8 | — | |
HWJADHWXPJWORQ
|
7.0 | IC50 | 8 | — | |
IXSNCCSCCZNQIN
|
7.0 | IC50 | 8 | — | |
LMUCVOYUWPGAFT
|
7.0 | IC50 | 8 | — | |
QBKNGTZPHDZTCI
|
7.0 | IC50 | 8 | — | |
XMLRYSWFMKXBFZ
|
7.0 | IC50 | 8 | — | |
JOGKUKXHTYWRGZ
|
7.0 | IC50 | 28 | — | |
YTYDCEPEGBYJIP
|
7.0 | IC50 | 8 | — | |
QBURVOCVNFVRQH
|
7.0 | IC50 | 8 | — | |
QGFAJQWXDUOVND
|
7.0 | IC50 | 8 | — |