Target Details
| UniProt AC | Q8WXS5 |
|---|---|
| Gene Symbol | CACNG8 |
| Protein Name | Voltage-dependent calcium channel gamma-8 subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00822 (PMP22_Claudin) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (7)
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AYAICAKEBFTALD
|
9.7 | IC50 | 2 | — | |
TWUDJPWCVJDVTM
|
8.7 | IC50 | 26 | — | |
CQCHOVDIAHVBMQ
|
8.7 | IC50 | 26 | — | |
LQNBSHGSEOTYDZ
|
8.6 | IC50 | 26 | — | |
BBGOPUNRXCQCNZ
|
8.6 | IC50 | 2 | — | |
FFERWAZVBAHCCT
|
8.6 | IC50 | 2 | — | |
UIHAKIQDNUUYNT
|
8.6 | IC50 | 2 | — | |
TYXGRJPOMQEXJV
|
8.5 | IC50 | 26 | — | |
GTVKXVAXHKIMQX
|
8.5 | IC50 | 26 | — | |
HACCLYCGUNUBJY
|
8.2 | IC50 | 26 | — | |
FRGPFJVINLDQIJ
|
8.2 | IC50 | 26 | — | |
JWZPZXKJEUAZFV
|
8.2 | IC50 | 26 | — | |
HQVBGHWQIKPZCY
|
8.2 | IC50 | 2 | — | |
RIAAESBLPRZGAK
|
8.2 | IC50 | 26 | — | |
AJCGCPQKWYQPNQ
|
8.1 | IC50 | 26 | — | |
DAMJJTRLEZYXQM
|
8.1 | IC50 | 26 | — | |
HNSMBMPEJNXIBA
|
8.1 | IC50 | 2 | — | |
QUYJROSEXGBONG
|
8.1 | IC50 | 26 | — | |
OXIUFIQCDNTAED
|
8.1 | IC50 | 26 | — | |
YEOAYGDVMJPHGG
|
8.0 | IC50 | 26 | — | |
OSYITGFTDTWGJW
|
8.0 | IC50 | 26 | — | |
COBXSLRIXGQVGS
|
8.0 | IC50 | 2 | — | |
WJCNWFPRVRWFCU
|
8.0 | IC50 | 2 | — | |
UGCISYLUHGKJKT
|
8.0 | IC50 | 26 | — | |
SRGBARMXFGWMTF
|
7.9 | IC50 | 26 | — | |
CNCRGRBWUATVCP
|
7.8 | IC50 | 26 | — | |
YZIYDQGNWSHQSD
|
7.8 | IC50 | 26 | — | |
ZMYGBEMRHGJETO
|
7.8 | IC50 | 26 | — | |
NOCIOWGNSBLDHC
|
7.8 | IC50 | 26 | — | |
NWSFHJWTWBRJFA
|
7.8 | IC50 | 26 | — | |
KDQVOHZGLRUPLF
|
7.8 | IC50 | 2 | — | |
CLSLOWKHEUDMRP
|
7.7 | IC50 | 26 | — | |
ZTNBOUBFOFURTR
|
7.6 | IC50 | 26 | — | |
BDMBSHGVIWYMFZ
|
7.6 | IC50 | 26 | — | |
BDZDJFPQRUGPOF
|
7.5 | IC50 | 26 | — | |
BVNRYPXFJUABAB
|
7.5 | IC50 | 26 | — | |
NRQIYYZXZYUWFB
|
7.5 | IC50 | 26 | — | |
VLKBVXIFTQLGCO
|
7.5 | IC50 | 26 | — | |
MVUOEDQURQKALH
|
7.5 | IC50 | 26 | — | |
PSVKDIGKMXLUQF
|
7.5 | IC50 | 26 | — | |
IXSXSOMMKYUETH
|
7.5 | IC50 | 26 | — | |
FFLKWIPCJQAAJX
|
7.4 | IC50 | 26 | — | |
QRGMHEOPAKSEPT
|
7.4 | IC50 | 26 | — | |
UMDPFCNSBNGNBU
|
7.4 | IC50 | 26 | — | |
QWTOYMMBYIZUDZ
|
7.4 | IC50 | 26 | — | |
DGLLVIVBOKDIKT
|
7.3 | IC50 | 2 | — | |
HXOISDVBEMOPLN
|
7.3 | IC50 | 2 | — | |
ZWJKOWFFHJCZRL
|
7.3 | IC50 | 26 | — | |
XNUZTIQWJMXUHN
|
7.2 | IC50 | 26 | — | |
AZSLSVQTOKQPLV
|
7.2 | IC50 | 26 | — |