Target Details
| UniProt AC | Q8WTQ7 |
|---|---|
| Gene Symbol | GRK7 |
| Protein Name | Rhodopsin kinase GRK7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 19
- Clinical molecules 9
- Avg pChEMBL 6.87
KEGG Pathways (3)
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.3 | IC50 | 408 | — | |
ACLLLJSNOCYQOJ
|
8.2 | IC50 | 8 | — | |
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
GYMOXCZIQHPXOH
|
7.8 | IC50 | 6 | — | |
PTJBMQVUHYZJLN
|
7.4 | IC50 | 5 | — | |
BMGQWWVMWDBQGC
|
7.3 | Kd | 147 | Yes | |
OYONTEXKYJZFHA
|
7.2 | Kd | 69 | Yes | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
XYUFCXJZFZPEJD
|
6.7 | IC50 | 23 | Yes | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
KGPGFQWBCSZGEL
|
6.4 | Kd | 59 | Yes | |
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
HFNKQEVNSGCOJV
|
6.3 | Kd | 65 | — | |
HZTYDQRUAWIZRE
|
6.3 | Kd | 40 | Yes | |
ZZSBPGIGIUFJRA
|
6.3 | Kd | 46 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
XQVVPGYIWAGRNI
|
6.1 | Kd | 34 | — | |
BIIVYFLTOXDAOV
|
6.0 | Kd | 82 | Yes |