Target Details
| UniProt AC | Q8WQX9 |
|---|---|
| Gene Symbol | PDEB1 |
| Protein Name | Phosphodiesterase |
| Organism | Trypanosoma brucei |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 68
- Clinical molecules 0
- Avg pChEMBL 6.84
Active Molecules (68)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QOKLLNXWXGSSRT
|
6.4 | Ki | 2 | — | |
RVULXXBAJKOFDU
|
6.4 | Ki | 2 | — | |
WVAQTVIALKSAMT
|
6.4 | Ki | 2 | — | |
LKXRSFQDUFXVGE
|
6.3 | Ki | 2 | — | |
LQRHIYIFVVRJJY
|
6.3 | Ki | 2 | — | |
PVSVGRCSLUMZQM
|
6.3 | Ki | 2 | — | |
DMGPHLQXDFXKSM
|
6.2 | Ki | 2 | — | |
KIILUOSGHLGYRG
|
6.2 | Kd | 3 | — | |
NPAQBDQEMKKBJM
|
6.2 | Ki | 2 | — | |
YALZXZYFCQHHIY
|
6.2 | Ki | 2 | — | |
FCHKQUZBYFBHFC
|
6.2 | Ki | 2 | — | |
JEGOZEYWJOCXNL
|
6.2 | Ki | 2 | — | |
BYDYPOWTTDVEFN
|
6.2 | Ki | 2 | — | |
FBGVWTSIULXAAQ
|
6.1 | Ki | 2 | — | |
XHVNSQNQZGAFGQ
|
6.1 | Ki | 2 | — | |
OGVVVHXXDFPPNX
|
6.0 | IC50 | 2 | — | |
BQEKCTABABAGDE
|
6.0 | Ki | 2 | — | |
FCFZXPZNUOXBMS
|
6.0 | Ki | 2 | — |