Target Details
| UniProt AC | Q8TF76 |
|---|---|
| Gene Symbol | HASPIN |
| Protein Name | Serine/threonine-protein kinase haspin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12330 (Haspin_kinase) |
Summary
- Multi-target molecules 103
- Clinical molecules 1
- Avg pChEMBL 7.13
Active Molecules (103)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTNDZQHUJGBYAQ
|
7.0 | IC50 | 4 | — | |
IRVDFMPPZOLHDV
|
7.0 | IC50 | 4 | — | |
YENIGUGPROEFFL
|
7.0 | IC50 | 3 | — | |
DMNJQOOMCYGQDB
|
6.9 | IC50 | 2 | — | |
PUALMDIOHBZAKU
|
6.9 | IC50 | 2 | — | |
MAJHBOYILMHFIY
|
6.9 | IC50 | 3 | — | |
RAXZSEGXMBWYQK
|
6.9 | Kd | 21 | — | |
IQJKHKMDUAVVBY
|
6.9 | IC50 | 4 | — | |
LVQICVKIHBQMRT
|
6.9 | IC50 | 4 | — | |
VAVPZKLEJFEUAP
|
6.8 | IC50 | 4 | — | |
FKSAHKFFMSBYIJ
|
6.8 | IC50 | 4 | — | |
FQBRQRVXPUQKLG
|
6.8 | IC50 | 4 | — | |
NXBHOGUUOJAZBN
|
6.8 | IC50 | 4 | — | |
UHXNWKPYFGCGQC
|
6.8 | IC50 | 3 | — | |
PTDBRIWRJGOEOL
|
6.8 | IC50 | 3 | — | |
HQJBUERUDFFUCK
|
6.7 | IC50 | 4 | — | |
KVXMBXJEXMWXLQ
|
6.7 | IC50 | 4 | — | |
KMJBSZNZTUBEMD
|
6.7 | IC50 | 4 | — | |
YRNKBHIBUTYIHE
|
6.7 | IC50 | 3 | — | |
PGQXYWLBZYAGCM
|
6.7 | IC50 | 4 | — | |
FNIZWTONUSWDQJ
|
6.7 | IC50 | 4 | — | |
AMPPIJHFLHITHG
|
6.6 | IC50 | 4 | — | |
WBHQPLISMLDBLH
|
6.6 | IC50 | 4 | — | |
HIHDNOVBJSCLBP
|
6.6 | IC50 | 4 | — | |
NWCRGOGGLIDBKF
|
6.6 | IC50 | 3 | — | |
OQLIIBOECZZXCB
|
6.6 | IC50 | 3 | — | |
YPHSCPUMUBJQTH
|
6.5 | IC50 | 3 | — | |
ZUODKONSNNHSAJ
|
6.5 | IC50 | 7 | — | |
FNIZWTONUSWDQJ
|
6.5 | IC50 | 4 | — | |
YWOFSCOHZWEQFW
|
6.5 | IC50 | 3 | — | |
BBKBILBUEYTDFO
|
6.5 | IC50 | 3 | — | |
TZFYFJYOXYWJIK
|
6.5 | IC50 | 4 | — | |
HDAJDNHIBCDLQF
|
6.5 | IC50 | 14 | — | |
ZICLKVKKMGHHDX
|
6.5 | IC50 | 4 | — | |
CEWROMVZNURIEF
|
6.5 | IC50 | 4 | — | |
QXGOBEONKUXLNG
|
6.4 | IC50 | 4 | — | |
KZKRLQXEKDKIKC
|
6.4 | IC50 | 3 | — | |
AWPWSWALRFFFFR
|
6.3 | IC50 | 2 | — | |
BMRRXZPZWHSZCA
|
6.3 | IC50 | 3 | — | |
HKXZWCYJOVYJAX
|
6.3 | IC50 | 3 | — | |
ACPOUJIDANTYHO
|
6.3 | IC50 | 17 | Yes | |
IRVDFMPPZOLHDV
|
6.3 | IC50 | 4 | — | |
BXNJHAXVSOCGBA
|
6.2 | IC50 | 14 | — | |
VLALJCBKWZZVIP
|
6.2 | IC50 | 4 | — | |
ZQRVIVRAYKMRTB
|
6.2 | IC50 | 3 | — | |
IZSOMURGNGNGOR
|
6.2 | IC50 | 4 | — | |
ZYDJMSALOSSIES
|
6.1 | IC50 | 3 | — | |
MKZPLFJRGIIGLE
|
6.1 | IC50 | 3 | — | |
SATMZMMKDDTOSQ
|
6.1 | IC50 | 2 | — | |
DFKOEXFVNULJFQ
|
6.1 | IC50 | 3 | — |