Target Details
| UniProt AC | Q8TF76 |
|---|---|
| Gene Symbol | HASPIN |
| Protein Name | Serine/threonine-protein kinase haspin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12330 (Haspin_kinase) |
Summary
- Multi-target molecules 103
- Clinical molecules 1
- Avg pChEMBL 7.13
Active Molecules (103)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IYNFVHYXEIOETE
|
10.3 | Kd | 2 | — | |
ZPQGOZNGTXPGAU
|
9.9 | Kd | 2 | — | |
DSWGFGIRFVKDCY
|
9.3 | Kd | 2 | — | |
CZZCAOGIEGXMBZ
|
8.7 | IC50 | 10 | — | |
OPIMPFVNTDPVQW
|
8.5 | IC50 | 2 | — | |
DJVYXMINSBMUHH
|
8.4 | IC50 | 8 | — | |
DJVYXMINSBMUHH
|
8.4 | IC50 | 8 | — | |
WHSIXKUPQCKWBY
|
8.3 | IC50 | 6 | — | |
BRIBVJICQJDZMF
|
8.3 | Kd | 2 | — | |
RRAVJRJCTBGPCG
|
8.1 | IC50 | 3 | — | |
FFNTZJOKBZFDQL
|
8.0 | IC50 | 4 | — | |
QXPHUXPNTWFKOR
|
8.0 | IC50 | 4 | — | |
ZFOMCSNUEHMROO
|
8.0 | IC50 | 7 | — | |
ZJKIGHOTHYACFW
|
8.0 | IC50 | 6 | — | |
KYQSFDSQEWSVRH
|
8.0 | Kd | 2 | — | |
MPEULGZDXWQEGW
|
7.9 | IC50 | 4 | — | |
YRFOQHHFWYWAST
|
7.9 | IC50 | 22 | — | |
IFLBFWBMAWIBBZ
|
7.8 | Kd | 7 | — | |
ITRXYWUAAUJIKA
|
7.8 | IC50 | 4 | — | |
LMVYGYMGJZTISD
|
7.8 | IC50 | 3 | — | |
YZQXGSFVWSAYFN
|
7.8 | IC50 | 3 | — | |
BIBOVMGNFAPEJA
|
7.7 | IC50 | 4 | — | |
AFQAFERZBGFZRQ
|
7.6 | IC50 | 4 | — | |
HIFKRZORZOSOFC
|
7.6 | IC50 | 4 | — | |
MXPUHLQPJSPPAS
|
7.6 | IC50 | 4 | — | |
YHBCYQIXVZFFIV
|
7.6 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.5 | IC50 | 408 | — | |
ZRCRKSJBXVRFPW
|
7.5 | IC50 | 4 | — | |
MHXGEROHKGDZGO
|
7.5 | IC50 | 10 | — | |
ISQMHRGAJWVQET
|
7.5 | IC50 | 4 | — | |
GLCIBEGENZSGCS
|
7.4 | IC50 | 3 | — | |
HAUGVIAEKSQIGA
|
7.4 | IC50 | 4 | — | |
ADNJUAOLUJJJHY
|
7.4 | IC50 | 4 | — | |
YSMNHYFBBOMUFX
|
7.4 | Kd | 3 | — | |
ZOOJEBLXLLZVIR
|
7.4 | IC50 | 4 | — | |
URTXFNMSFMYZRA
|
7.4 | IC50 | 4 | — | |
FSBMCTDYWXIBLM
|
7.3 | IC50 | 22 | — | |
IVMAILZOXLZXTB
|
7.3 | IC50 | 4 | — | |
KOZWDURZSCBPDP
|
7.3 | IC50 | 4 | — | |
NFFNNAYVKWIBSG
|
7.3 | IC50 | 4 | — | |
WPPGBVWZGMDXKF
|
7.2 | IC50 | 5 | — | |
XHVYRNHFNKLZPA
|
7.1 | IC50 | 4 | — | |
DFIYULDPYGDCHT
|
7.1 | IC50 | 2 | — | |
FUSZCAJFRIHBLV
|
7.1 | IC50 | 4 | — | |
UHSYUXJDTQLOMQ
|
7.1 | IC50 | 3 | — | |
NBJYPTQHFDBQQA
|
7.1 | IC50 | 3 | — | |
TTXDQGLSSNHEQI
|
7.1 | IC50 | 4 | — | |
NENJFZKQHYXRDQ
|
7.1 | Kd | 8 | — | |
ZPUYWMRULPSNOR
|
7.1 | IC50 | 4 | — | |
ZHJUEEVXBXXRCT
|
7.0 | IC50 | 4 | — |