Target Details
| UniProt AC | Q8TDC3 |
|---|---|
| Gene Symbol | BRSK1 |
| Protein Name | Serine/threonine-protein kinase BRSK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21122 (KA1_BRSK) PF00069 (Pkinase) PF21115 (UBA_BRSK) |
Summary
- Multi-target molecules 70
- Clinical molecules 8
- Avg pChEMBL 6.67
Active Molecules (70)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MLGGUGPIWDHBAI
|
6.2 | Ki | 33 | — | |
PNAPQQCRNHMIER
|
6.2 | Ki | 12 | — | |
QNUKRWAIZMBVCU
|
6.2 | Ki | 46 | — | |
SHENEEFOURUIBP
|
6.2 | Ki | 29 | — | |
WYOMXSAYYXBPMN
|
6.2 | Ki | 24 | — | |
YMIJUBCSOKSFRU
|
6.2 | Ki | 87 | — | |
UJIAQDJKSXQLIT
|
6.1 | Kd | 38 | — | |
AOBLBPWPSKBHSI
|
6.1 | Ki | 55 | — | |
GCBJDOWIQHMCMR
|
6.1 | Ki | 84 | — | |
KRIUNPBAQZGFQA
|
6.1 | Ki | 76 | — | |
PSCJSWRVCKUMSL
|
6.1 | Ki | 35 | — | |
UYJNQQDJUOUFQJ
|
6.1 | Ki | 68 | — | |
WVFWTUJEHMVUBG
|
6.1 | Ki | 25 | — | |
DKXHSOUZPMHNIZ
|
6.0 | Ki | 51 | Yes | |
FUMCKNCUEAQHCV
|
6.0 | Ki | 103 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
OLVBAUVSICCWEJ
|
6.0 | Ki | 39 | — | |
PTVPBWWDGZSEAF
|
6.0 | Ki | 63 | — |