Target Details
| UniProt AC | Q8TDC3 |
|---|---|
| Gene Symbol | BRSK1 |
| Protein Name | Serine/threonine-protein kinase BRSK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21122 (KA1_BRSK) PF00069 (Pkinase) PF21115 (UBA_BRSK) |
Summary
- Multi-target molecules 70
- Clinical molecules 8
- Avg pChEMBL 6.67
Active Molecules (70)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.9 | IC50 | 408 | — | |
JLWGOAGEDWMEBT
|
8.7 | IC50 | 10 | — | |
JLWGOAGEDWMEBT
|
8.7 | IC50 | 10 | — | |
GCYXEGSPUDSZJY
|
7.9 | Ki | 82 | — | |
MFAQYJIYDMLAIM
|
7.8 | Kd | 130 | Yes | |
CZIGMBNEFWBEMD
|
7.6 | Ki | 16 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
KWRXWPRFIUJQBP
|
7.5 | Ki | 25 | — | |
OWRXHGAFWZFFCW
|
7.4 | Ki | 113 | — | |
RJZDECGDCKOHBV
|
7.4 | Ki | 70 | — | |
NZVDDFRUBIEKLV
|
7.3 | Ki | 20 | — | |
AWDORCFLUJZUQS
|
7.1 | Ki | 22 | — | |
LRZYYIZFBXFSJB
|
7.1 | Ki | 69 | — | |
RYYNGWLOYLRZLK
|
7.1 | Ki | 104 | — | |
VUHZDNOPEVGHEO
|
7.1 | Ki | 29 | — | |
ZKHDDJKHTPLPOQ
|
7.1 | Ki | 62 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
AZTMYWWWILJAKW
|
6.9 | Ki | 16 | Yes | |
BSFNGHCTZDCQBF
|
6.8 | Ki | 93 | — | |
DFMCXVONDDGQIY
|
6.8 | Ki | 66 | — | |
OLUKILHGKRVDCT
|
6.8 | Ki | 44 | Yes | |
QPORZABOFXPRHM
|
6.8 | Ki | 18 | — | |
WINHZLLDWRZWRT
|
6.8 | Ki | 66 | — | |
CMWRPDHVGMHLSZ
|
6.7 | IC50 | 22 | — | |
OSVUGUHRKMMBSE
|
6.7 | Kd | 170 | — | |
MIKAKZKNMYZLDX
|
6.7 | Ki | 42 | — | |
RIBBPSYZBQQTQC
|
6.7 | Ki | 15 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
JAMDNXUAYUHJLJ
|
6.6 | Ki | 40 | — | |
JSKUWFIZUALZLX
|
6.6 | Ki | 33 | — | |
RITAVMQDGBJQJZ
|
6.6 | Ki | 33 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
CKVWQORGCCEYHS
|
6.5 | Ki | 50 | — | |
AILRADAXUVEEIR
|
6.5 | IC50 | 75 | — | |
AIQDZMUPVYDVLB
|
6.4 | Ki | 48 | — | |
PIQCTGMSNWUMAF
|
6.4 | Ki | 137 | Yes | |
QTQUAHGXBLFSCH
|
6.4 | Ki | 10 | — | |
XKFTZKGMDDZMJI
|
6.4 | Ki | 56 | — | |
XYZNKCSDQRKAFR
|
6.4 | Ki | 53 | — | |
GHPFSYCYZJKVDZ
|
6.3 | Ki | 18 | Yes | |
IAKGNUWZPSPEKU
|
6.3 | Ki | 19 | — | |
NHFDRBXTEDBWCZ
|
6.3 | Ki | 41 | — | |
NLUPJKQOKWBWFC
|
6.3 | Ki | 69 | — | |
UTFXYGYVDDLJER
|
6.3 | Ki | 36 | — | |
CXBBWVXSZINRCS
|
6.2 | Ki | 41 | — | |
FLEAYYMORDPWAJ
|
6.2 | Ki | 90 | — | |
GDYZFFBMSBDTAA
|
6.2 | Ki | 60 | — | |
HHSVICUMCOBRPT
|
6.2 | Ki | 33 | — | |
LRINYHMQZRENCY
|
6.2 | Ki | 29 | — |