Target Details
| UniProt AC | Q8TD19 |
|---|---|
| Gene Symbol | NEK9 |
| Protein Name | Serine/threonine-protein kinase Nek9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF25390 (WD40_RLD) |
Summary
- Multi-target molecules 18
- Clinical molecules 2
- Avg pChEMBL 6.61
Associated Diseases (2)
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHHQJBCNYHBUSI
|
7.8 | Kd | 220 | — | |
MWKSRKSEWLRPBL
|
7.6 | Kd | 1075 | — | |
GKDRMWXFWHEQQT
|
7.4 | Kd | 7 | — | |
BFSMGDJOXZAERB
|
7.3 | Kd | 33 | — | |
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
HKSZLNNOFSGOKW
|
7.0 | IC50 | 408 | — | |
JOOXLOJCABQBSG
|
6.8 | Kd | 139 | — | |
ZXNSGRMQSJUSGX
|
6.4 | Kd | 3 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
YYLKKYCXAOBSRM
|
6.3 | Kd | 191 | — | |
WVXNSAVVKYZVOE
|
6.2 | IC50 | 92 | — | |
LQVXSNNAFNGRAH
|
6.2 | Kd | 33 | Yes | |
KTEIFNKAUNYNJU
|
6.1 | Kd | 114 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |