Target Details
| UniProt AC | Q8TD08 |
|---|---|
| Gene Symbol | MAPK15 |
| Protein Name | Mitogen-activated protein kinase 15 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 42
- Clinical molecules 9
- Avg pChEMBL 6.92
KEGG Pathways (1)
Active Molecules (42)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
MCUJKPPARUPFJM
|
8.3 | Kd | 11 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
MWKSRKSEWLRPBL
|
7.7 | Kd | 1075 | — | |
RAXZSEGXMBWYQK
|
7.5 | Kd | 21 | — | |
RPGZQOOZHIEPJW
|
7.5 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.5 | Kd | 18 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
MLDQJTXFUGDVEO
|
7.3 | Kd | 85 | Yes | |
YRFOQHHFWYWAST
|
7.2 | IC50 | 22 | — | |
JRNJNYBQQYBCLE
|
7.2 | Kd | 40 | Yes | |
CXQHYVUVSFXTMY
|
7.1 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.1 | Kd | 149 | — | |
AXRCEOKUDYDWLF
|
7.1 | Kd | 31 | — | |
ZCBUQCWBWNUWSU
|
7.1 | Kd | 59 | — | |
BPNUQXPIQBZCMR
|
7.0 | Kd | 83 | Yes | |
DKZYXHCYPUVGAF
|
7.0 | Kd | 112 | — | |
ODPGGGTTYSGTGO
|
7.0 | Kd | 153 | — | |
XPYOCUNKDACBLQ
|
7.0 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
OUSFTKFNBAZUKL
|
6.9 | Kd | 58 | Yes | |
OVPNQJVDAFNBDN
|
6.9 | Kd | 44 | Yes | |
YBYYWUUUGCNAHQ
|
6.9 | IC50 | 8 | — | |
KOZFSFOOLUUIGY
|
6.8 | Kd | 88 | Yes | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
HUXYBQXJVXOMKX
|
6.6 | Kd | 28 | — | |
CVWXJKQAOSCOAB
|
6.6 | Kd | 35 | — | |
WVXNSAVVKYZVOE
|
6.6 | Kd | 92 | — | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
BIIVYFLTOXDAOV
|
6.5 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.5 | Kd | 82 | Yes | |
KRIWIRSMQRQYJG
|
6.5 | IC50 | 11 | — | |
YFBPGSDPFRCNOY
|
6.4 | IC50 | 2 | — | |
PMDAVRLCSZSLRH
|
6.4 | Kd | 13 | — | |
JOOXLOJCABQBSG
|
6.3 | Kd | 139 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
NXWXUDHOUKWAQU
|
6.2 | Kd | 16 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
XCOSAQGGGZDYJN
|
6.0 | IC50 | 11 | — |