Target Details
| UniProt AC | Q8TCW9 |
|---|---|
| Gene Symbol | PROKR1 |
| Protein Name | Prokineticin receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 70
- Clinical molecules 0
- Avg pChEMBL 6.57
Active Molecules (70)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OROHKZMWESPHLN
|
8.6 | Ki | 2 | — | |
STQKBSSAMXUHBU
|
8.6 | Ki | 2 | — | |
AJYKZRXAHQYRHZ
|
8.4 | Ki | 2 | — | |
QGZNVUJOSDSAHH
|
8.1 | Ki | 2 | — | |
FKOOTUPWQZIUKE
|
7.4 | IC50 | 2 | — | |
YZLYZJPLSNEUDJ
|
7.4 | IC50 | 2 | — | |
HHEXKHCZHUFGSZ
|
7.3 | IC50 | 2 | — | |
HIPWXCNVKOZTAR
|
7.3 | IC50 | 2 | — | |
HGWURKAPEFTTEO
|
7.2 | IC50 | 2 | — | |
JTGYOXKVMCWCBO
|
7.2 | IC50 | 2 | — | |
ZUYOQHBOAKWQHG
|
7.2 | IC50 | 2 | — | |
OHMCLGXQLDFMFC
|
7.0 | Ki | 2 | — | |
OSRKPRHWTFIMHG
|
7.0 | IC50 | 2 | — | |
BYDVQJXWMGECPM
|
6.8 | IC50 | 2 | — | |
KRQZAVUNAGZXQM
|
6.8 | IC50 | 2 | — | |
HQZXREKXJOEQFU
|
6.8 | IC50 | 2 | — | |
BWNLVZDGPGZWRA
|
6.8 | IC50 | 2 | — | |
CSSWRQHXWZZJPC
|
6.8 | IC50 | 2 | — | |
UHEABFFWWVYGMU
|
6.8 | IC50 | 2 | — | |
YAXYBAJRIAAJBG
|
6.7 | IC50 | 2 | — | |
WDYRJTUJRWNENR
|
6.7 | IC50 | 2 | — | |
YBHHRLALVLWHFL
|
6.7 | IC50 | 2 | — | |
FKPHYHMWXCZHQK
|
6.7 | IC50 | 2 | — | |
HCVXGWGKJCDLHW
|
6.7 | IC50 | 2 | — | |
ORLKIYKAPSAHTN
|
6.7 | IC50 | 2 | — | |
AQGCEEFKPPNGMT
|
6.7 | IC50 | 2 | — | |
LVAYTVXWKWKIQK
|
6.6 | IC50 | 2 | — | |
LYHMQCQUGJIVRF
|
6.6 | IC50 | 2 | — | |
ZQNZGINXIFNSSP
|
6.5 | IC50 | 2 | — | |
YJHPFQHKOBNEJT
|
6.5 | IC50 | 2 | — | |
KSXBFKHWLTYGHZ
|
6.5 | IC50 | 2 | — | |
GLCNBMLOJYQRAF
|
6.5 | IC50 | 2 | — | |
QLIJDSZWYAYKRZ
|
6.4 | IC50 | 2 | — | |
JDTHPTFPMSSAJL
|
6.4 | IC50 | 2 | — | |
AXYFHHUNIHMJGQ
|
6.4 | IC50 | 2 | — | |
AYWHPILLEOWBLQ
|
6.4 | IC50 | 2 | — | |
MKOGIKITDSUWCY
|
6.3 | IC50 | 2 | — | |
OLSSEGPWHBZHOA
|
6.3 | IC50 | 2 | — | |
UHAAKMVWUJVWNK
|
6.3 | IC50 | 2 | — | |
VIAFMEZYCPFRJF
|
6.3 | IC50 | 2 | — | |
GYDNBJRNRTVGET
|
6.3 | IC50 | 2 | — | |
KJERPMGHBIDYES
|
6.3 | IC50 | 2 | — | |
ROCOKNRCXBAIJD
|
6.3 | IC50 | 2 | — | |
ZNJXCUJSFQGQJE
|
6.3 | IC50 | 2 | — | |
BPOFQMPOUZNIFN
|
6.3 | IC50 | 2 | — | |
NSVJNZFPHAVCDE
|
6.2 | IC50 | 2 | — | |
RCJMVXOOADTNLX
|
6.2 | IC50 | 2 | — | |
FHILMZDTYLGGMQ
|
6.2 | IC50 | 2 | — | |
QNHZGRPXIDABBQ
|
6.2 | IC50 | 2 | — | |
UWMGWHFTRQZUNM
|
6.2 | IC50 | 2 | — |