Target Details
| UniProt AC | Q8TBC4 |
|---|---|
| Gene Symbol | UBA3 |
| Protein Name | NEDD8-activating enzyme E1 catalytic subunit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08825 (E2_bind) PF00899 (ThiF) |
Summary
- Multi-target molecules 127
- Clinical molecules 0
- Avg pChEMBL 7.01
KEGG Pathways (1)
Active Molecules (127)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBPMFDHRGACICG
|
6.9 | IC50 | 2 | — | |
MUJHZPSIEOHDFE
|
6.9 | IC50 | 4 | — | |
IFIIGJXRDOYWOO
|
6.8 | IC50 | 2 | — | |
VOUGYOLBJNTWOJ
|
6.8 | IC50 | 2 | — | |
UHZSMEDUPPKHQT
|
6.8 | IC50 | 2 | — | |
CSHUTMOBESIZLB
|
6.7 | IC50 | 2 | — | |
KIDRXSDFGBELIZ
|
6.7 | IC50 | 4 | — | |
HKKCQZRJLCIYQD
|
6.7 | IC50 | 4 | — | |
QGKYPQQBUWTDAI
|
6.7 | IC50 | 4 | — | |
HVYXBVYVVDINDV
|
6.7 | IC50 | 2 | — | |
UKXNNPGADCVLBH
|
6.7 | IC50 | 4 | — | |
RCFBEFLWLRKPSK
|
6.7 | IC50 | 2 | — | |
PZCKLTWSXFDLLP
|
6.6 | IC50 | 6 | — | |
JMXCOZRAISPELW
|
6.6 | IC50 | 4 | — | |
SDTFURRUMBVNTO
|
6.6 | IC50 | 4 | — | |
DQGFFQCTFTZJDD
|
6.6 | IC50 | 4 | — | |
ZHYGWRCVOBRNRJ
|
6.6 | IC50 | 4 | — | |
WYUXXLIVBAVLGU
|
6.6 | IC50 | 4 | — | |
KJNKXIWPYBQGTE
|
6.5 | IC50 | 4 | — | |
IXCWIEAIJGSNQZ
|
6.5 | IC50 | 4 | — | |
SPZOHGTXTGPSCS
|
6.5 | IC50 | 4 | — | |
XYUKAKFBAWCQRY
|
6.5 | IC50 | 4 | — | |
SCHCQZKKFVETHG
|
6.5 | IC50 | 4 | — | |
XRTNAEKEDZVZHF
|
6.5 | IC50 | 4 | — | |
MCVBNJJPKVQNHA
|
6.5 | IC50 | 4 | — | |
OMEJZYALSBXTSP
|
6.5 | IC50 | 4 | — | |
PJHUELIKSXLGBB
|
6.5 | IC50 | 4 | — | |
HKIARJIHQHADQP
|
6.4 | IC50 | 6 | — | |
CEHPNXFEKRRQBD
|
6.4 | IC50 | 4 | — | |
IMAHPWNULQNTBO
|
6.3 | IC50 | 4 | — | |
RZAVZYBRGRFZIG
|
6.3 | IC50 | 4 | — | |
AHKKODSOFUTMPM
|
6.3 | IC50 | 2 | — | |
CLKAMYMBIRKTSG
|
6.3 | IC50 | 2 | — | |
DMAKVCMEOOHYAB
|
6.3 | IC50 | 2 | — | |
FLMZTLYOGVPHDB
|
6.3 | IC50 | 2 | — | |
FTQUIPPXVTVAKQ
|
6.3 | IC50 | 2 | — | |
GUKGTVMKUPBWOJ
|
6.3 | IC50 | 2 | — | |
HHMPQFVUXYKGLH
|
6.3 | IC50 | 2 | — | |
HHMPQFVUXYKGLH
|
6.3 | IC50 | 2 | — | |
HRSCTJKWHYEIEF
|
6.3 | IC50 | 2 | — | |
HSXWEADXTURRPO
|
6.3 | IC50 | 2 | — | |
IINUZRFVTDDCRA
|
6.3 | IC50 | 2 | — | |
IOYFJTJXBYRHPS
|
6.3 | IC50 | 2 | — | |
IWOWZEOZEPKONU
|
6.3 | IC50 | 2 | — | |
IWOWZEOZEPKONU
|
6.3 | IC50 | 2 | — | |
IXADUWXIFADGDC
|
6.3 | IC50 | 2 | — | |
KFKCYVLWIBQJFZ
|
6.3 | IC50 | 2 | — | |
KVFDWIYTEKHZET
|
6.3 | IC50 | 2 | — | |
KXEDUHGELOKWOR
|
6.3 | IC50 | 2 | — | |
KXEDUHGELOKWOR
|
6.3 | IC50 | 2 | — |