Target Details
| UniProt AC | Q8T6T2 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Inosine-5'-monophosphate dehydrogenase |
| Organism | Cryptosporidium parvum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00478 (IMPDH) |
Summary
- Multi-target molecules 26
- Clinical molecules 0
- Avg pChEMBL 7.51
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUFRXADFMZVJFT
|
9.2 | IC50 | 2 | — | |
IMBVKBZWLRXRAW
|
9.1 | IC50 | 2 | — | |
LORXIJMHWYBXHQ
|
9.0 | IC50 | 2 | — | |
HRXGXBGJVNUGSX
|
8.7 | IC50 | 2 | — | |
NTLVMPJCDHOJPI
|
8.4 | IC50 | 2 | — | |
NRJRCKIOCQMNMC
|
8.3 | Ki | 2 | — | |
QCNXGTHMVPSAAC
|
8.0 | IC50 | 2 | — | |
DSTKQECXQMKQLN
|
7.9 | Ki | 2 | — | |
XYCMWFINXXFAFG
|
7.9 | IC50 | 2 | — | |
TYHBRTURECWDPC
|
7.8 | Ki | 2 | — | |
GMQDVIPGHXODOQ
|
7.5 | IC50 | 2 | — | |
HLCZIGFLGPKWJH
|
7.4 | Ki | 2 | — | |
XDGYRLMYUQCESN
|
7.4 | Ki | 2 | — | |
GEIJWCQHHWUHNK
|
7.4 | Ki | 2 | — | |
GFKRWPNMQSLPGF
|
7.3 | Ki | 2 | — | |
PWBTYBHLXLDUDX
|
7.3 | IC50 | 2 | — | |
KJTBISSTZHKHKQ
|
7.2 | Ki | 2 | — | |
UEIJVWKUAHOKDQ
|
7.2 | Ki | 2 | — | |
MSWDVKDZSZKCSP
|
7.0 | Ki | 2 | — | |
UYWWATMWRMNMPI
|
6.9 | Ki | 2 | — | |
NGENHIWQQFTCNF
|
6.8 | Ki | 2 | — | |
ZOPVXVNGASGEIR
|
6.7 | IC50 | 2 | — | |
UMSBQBXESMWNSM
|
6.5 | IC50 | 2 | — | |
NGENHIWQQFTCNF
|
6.3 | Ki | 2 | — | |
QZKIXDSVUHUHBH
|
6.2 | IC50 | 2 | — | |
BHWCXEGEAIORHG
|
6.0 | IC50 | 2 | — |