Target Details
| UniProt AC | Q8NFU7 |
|---|---|
| Gene Symbol | TET1 |
| Protein Name | Methylcytosine dioxygenase TET1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12851 (Tet_JBP) PF02008 (zf-CXXC) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 6.47
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RYSZEZFKNLPKJY
|
7.2 | IC50 | 3 | — | |
JWDOHVSTMORFKO
|
6.6 | IC50 | 2 | — | |
QPAVDBKPIQERNE
|
6.6 | IC50 | 2 | — | |
JHBMFEYJXZTCEA
|
6.4 | IC50 | 3 | — | |
OTEYSQVKIKPKFX
|
6.2 | IC50 | 3 | — | |
JGRPKOGHYBAVMW
|
6.2 | IC50 | 13 | — | |
RXNGLDYXFDNFEX
|
6.1 | IC50 | 2 | — |