Target Details
| UniProt AC | Q8NFD2 |
|---|---|
| Gene Symbol | ANKK1 |
| Protein Name | Ankyrin repeat and protein kinase domain-containing protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 16
- Clinical molecules 5
- Avg pChEMBL 6.48
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
PIQCTGMSNWUMAF
|
7.1 | Kd | 137 | Yes | |
YYLKKYCXAOBSRM
|
7.1 | Kd | 191 | — | |
CTNPALGJUAXMMC
|
6.8 | Kd | 151 | — | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 213 | — | |
WINHZLLDWRZWRT
|
6.5 | Kd | 201 | Yes | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
HFNKQEVNSGCOJV
|
6.4 | Kd | 65 | — | |
KDKUVYLMPJIGKA
|
6.3 | Kd | 91 | Yes | |
ODPGGGTTYSGTGO
|
6.2 | Kd | 153 | — | |
KTEIFNKAUNYNJU
|
6.1 | Kd | 114 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MVCOAUNKQVWQHZ
|
6.0 | Kd | 54 | Yes |