Target Details
| UniProt AC | Q8NE63 |
|---|---|
| Gene Symbol | HIPK4 |
| Protein Name | Homeodomain-interacting protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 183
- Clinical molecules 26
- Avg pChEMBL 6.83
KEGG Pathways (1)
Active Molecules (183)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ISVHLTLEHRZKJC
|
6.2 | Ki | 19 | — | |
JJJSCYSPSKBQAX
|
6.2 | Ki | 34 | — | |
MTYMWGNJKDHWGN
|
6.2 | Ki | 18 | — | |
RAPYFGJGASETOS
|
6.2 | Ki | 11 | — | |
ZLVOTRRGLSDLPF
|
6.2 | Ki | 36 | — | |
SVNVPNHWFJFRLZ
|
6.2 | IC50 | 8 | — | |
BPNUQXPIQBZCMR
|
6.1 | Kd | 83 | Yes | |
FAIHBCXQSBIRIL
|
6.1 | Ki | 22 | — | |
FLEAYYMORDPWAJ
|
6.1 | Ki | 90 | — | |
HHSVICUMCOBRPT
|
6.1 | Ki | 33 | — | |
JRVSFZKYQCETAH
|
6.1 | Ki | 19 | — | |
OWDRQHVEJIYVOI
|
6.1 | Ki | 47 | — | |
TZSJMSZEKQGCBI
|
6.1 | Ki | 15 | — | |
VUHZDNOPEVGHEO
|
6.1 | Ki | 29 | — | |
AAKJLRGGTJKAMG
|
6.0 | Kd | 50 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 147 | Yes | |
KTUFNOKKBVMGRW
|
6.0 | Kd | 38 | Yes | |
CTNPALGJUAXMMC
|
6.0 | Kd | 151 | — | |
HCNIBOQWDVOZKF
|
6.0 | Ki | 26 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JAMDNXUAYUHJLJ
|
6.0 | Ki | 40 | — | |
KAICHBSRWFIESE
|
6.0 | Ki | 14 | — | |
KHOVFNRAIYTEPO
|
6.0 | Ki | 5 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
OUJZYQBEFNDJQN
|
6.0 | Ki | 71 | — | |
VBUWAJWPXASNGM
|
6.0 | Ki | 9 | — | |
VNGYQBMDQMDALH
|
6.0 | Ki | 25 | — | |
XSRHBCYNCKAFKS
|
6.0 | Ki | 45 | — | |
YYLKKYCXAOBSRM
|
6.0 | Kd | 191 | — | |
ZGZVRPRSFXRGCF
|
6.0 | Ki | 76 | — | |
ZKHDDJKHTPLPOQ
|
6.0 | Ki | 62 | — | |
ZVWRFVCNQOECJS
|
6.0 | Ki | 71 | — |