Target Details
| UniProt AC | Q8NE63 |
|---|---|
| Gene Symbol | HIPK4 |
| Protein Name | Homeodomain-interacting protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 183
- Clinical molecules 26
- Avg pChEMBL 6.83
KEGG Pathways (1)
Active Molecules (183)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOBLBPWPSKBHSI
|
6.5 | Ki | 55 | — | |
CNTCGRJDUJEUDG
|
6.5 | Ki | 37 | — | |
CVWXJKQAOSCOAB
|
6.5 | Kd | 35 | — | |
GHAZVJQMLWOQLP
|
6.5 | Ki | 17 | — | |
GUMBHNMWKMFKRT
|
6.5 | Ki | 23 | — | |
HKSZLNNOFSGOKW
|
6.5 | IC50 | 408 | — | |
LCKDESRGCHSHHO
|
6.5 | Ki | 18 | — | |
PYXQMJSGJIJHJT
|
6.5 | Ki | 28 | — | |
RVSKJUNTDGBSSS
|
6.5 | Ki | 25 | — | |
XHORJSJFHVABEA
|
6.5 | Ki | 49 | — | |
XKZQZMSAWVDRSP
|
6.5 | Ki | 39 | Yes | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
ULXXDDBFHOBEHA
|
6.4 | Kd | 15 | Yes | |
FUMCKNCUEAQHCV
|
6.4 | Ki | 103 | — | |
GDYZFFBMSBDTAA
|
6.4 | Ki | 60 | — | |
GPKQGYSDQQIJLW
|
6.4 | Ki | 19 | — | |
HOBMVEVXDIOMDM
|
6.4 | Ki | 18 | — | |
IMHKMKWSWHFKTM
|
6.4 | Ki | 13 | — | |
OADRBDVURCEKRP
|
6.4 | Ki | 44 | — | |
OWFXKTOLFUQPDJ
|
6.4 | Ki | 36 | — | |
QAJPIJHWTGPUNZ
|
6.4 | Ki | 37 | — | |
RIUZPIBUSOHUKF
|
6.4 | Ki | 23 | — | |
RKUKAACYUCUJEE
|
6.4 | Ki | 58 | — | |
SVUIYNKSDCANAY
|
6.4 | Ki | 16 | — | |
UXXQOJXBIDBUAC
|
6.4 | Kd | 21 | Yes | |
XBYVOPRDASFDMY
|
6.4 | Ki | 42 | — | |
XFWUTMHVDGPWLH
|
6.4 | Ki | 75 | — | |
ZCXXFPLQFFRMPN
|
6.4 | Ki | 12 | — | |
NXSJMRCTGYTSTK
|
6.4 | Kd | 200 | — | |
WVXNSAVVKYZVOE
|
6.3 | IC50 | 92 | — | |
OSVUGUHRKMMBSE
|
6.3 | Kd | 170 | — | |
BIKYDWLMTPRSQL
|
6.3 | Ki | 50 | — | |
CKVWQORGCCEYHS
|
6.3 | Ki | 50 | — | |
IAKGNUWZPSPEKU
|
6.3 | Ki | 19 | — | |
KWRXWPRFIUJQBP
|
6.3 | Ki | 25 | — | |
LRLDYTTWQIFWBD
|
6.3 | Ki | 25 | — | |
LRZYYIZFBXFSJB
|
6.3 | Ki | 69 | — | |
MIKAKZKNMYZLDX
|
6.3 | Ki | 42 | — | |
MZDKLVOWGIOKTN
|
6.3 | Ki | 80 | — | |
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
TVEREFRWBLRPPJ
|
6.3 | Ki | 15 | — | |
XAYDUCQADQTDGX
|
6.3 | Ki | 12 | — | |
YWTBGJGMTBHQTM
|
6.3 | Ki | 65 | — | |
ZGDSBEUMPIMXBM
|
6.3 | Ki | 42 | — | |
VBYGXNURPHQSPG
|
6.3 | IC50 | 5 | — | |
YABJJWZLRMPFSI
|
6.2 | Kd | 34 | — | |
CHQYAWLKOUOTQO
|
6.2 | IC50 | 20 | — | |
ASNQMAVHHGGQRB
|
6.2 | Ki | 14 | — | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
DKXHSOUZPMHNIZ
|
6.2 | Ki | 51 | Yes |