Target Details
| UniProt AC | Q8NE63 |
|---|---|
| Gene Symbol | HIPK4 |
| Protein Name | Homeodomain-interacting protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 183
- Clinical molecules 26
- Avg pChEMBL 6.83
KEGG Pathways (1)
Active Molecules (183)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKZKELVPGXJIMW
|
7.1 | Ki | 41 | — | |
HRZOUBQYVUXBNS
|
7.1 | Ki | 38 | — | |
NLUPJKQOKWBWFC
|
7.1 | Ki | 69 | — | |
OUORNBBPANSKFS
|
7.1 | Ki | 3 | — | |
VCSQVKQFGYRGEH
|
7.1 | Ki | 13 | — | |
XLFYOIVELARSKP
|
7.1 | Ki | 33 | — | |
QYZOGCMHVIGURT
|
7.0 | Kd | 26 | Yes | |
CXQHYVUVSFXTMY
|
7.0 | IC50 | 154 | — | |
GEGCXGMFUYJULA
|
7.0 | Ki | 30 | Yes | |
MVJMMLFMPWITEJ
|
7.0 | Ki | 110 | — | |
OYONTEXKYJZFHA
|
7.0 | IC50 | 69 | Yes | |
QKPLUKMJEKRAJD
|
7.0 | Ki | 30 | Yes | |
SPMHGQZFMNZCBV
|
7.0 | Ki | 30 | Yes | |
UYJNQQDJUOUFQJ
|
7.0 | Ki | 68 | — | |
XYZNKCSDQRKAFR
|
7.0 | Ki | 53 | — | |
YEHCNYAQEBQCCS
|
7.0 | Ki | 74 | — | |
ZCBUQCWBWNUWSU
|
7.0 | IC50 | 59 | — | |
GMYYMEOGFRKSFS
|
6.9 | Ki | 29 | — | |
GQLWKGVBOIYMTN
|
6.9 | Ki | 35 | — | |
MULNSLQVKKUPJN
|
6.9 | Ki | 41 | — | |
RYAVJHIPOWNWDE
|
6.9 | Ki | 38 | — | |
UDFDIIVNIYWXDM
|
6.9 | Ki | 74 | — | |
UWDBNTXEKYRMSG
|
6.9 | Ki | 26 | — | |
WPXVVAWAHQHJPF
|
6.9 | IC50 | 41 | — | |
WVFWTUJEHMVUBG
|
6.9 | Ki | 25 | — | |
UBPYILGKFZZVDX
|
6.9 | Kd | 130 | Yes | |
UIARLYUEJFELEN
|
6.8 | Kd | 289 | Yes | |
GQHMZZXJWGPHDA
|
6.8 | Ki | 20 | — | |
LYNBNVBMAGDJRW
|
6.8 | Ki | 81 | — | |
MADCXGNPDBWPLM
|
6.8 | Ki | 25 | — | |
MTCHQDWUHQADSY
|
6.8 | Ki | 29 | — | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
WKEYMNLZBZKLOG
|
6.8 | Ki | 14 | — | |
WLKJMISWXHORCR
|
6.8 | IC50 | 11 | — | |
MJCKUHBSAUHVJE
|
6.7 | Ki | 4 | — | |
SOVYWBOZOBVFLP
|
6.7 | Ki | 10 | — | |
SPOBBSBKXJKGBG
|
6.7 | Ki | 16 | — | |
YEPNVBNYCRGZRX
|
6.7 | Ki | 26 | — | |
JOOXLOJCABQBSG
|
6.7 | Kd | 139 | — | |
CQBBMNXXVMOFCA
|
6.6 | Ki | 39 | — | |
IZAVTOABECKIDH
|
6.6 | Ki | 20 | — | |
KTQYQHLIMZOBSM
|
6.6 | Ki | 12 | — | |
LVECPYVAIBNSRV
|
6.6 | Ki | 33 | — | |
MHCPAORAYMTGCZ
|
6.6 | Ki | 37 | — | |
RJZDECGDCKOHBV
|
6.6 | Ki | 70 | — | |
WYOMXSAYYXBPMN
|
6.6 | Ki | 24 | — | |
YEKVTSRZMPLPFK
|
6.6 | Ki | 17 | — | |
RRIRDIKTUQVZCW
|
6.5 | Kd | 2 | — | |
XGALLCVXEZPNRQ
|
6.5 | Kd | 39 | Yes | |
ADLPKFFMGIJZIM
|
6.5 | Ki | 44 | — |