Target Details
| UniProt AC | Q8NE63 |
|---|---|
| Gene Symbol | HIPK4 |
| Protein Name | Homeodomain-interacting protein kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 183
- Clinical molecules 26
- Avg pChEMBL 6.83
KEGG Pathways (1)
Active Molecules (183)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEJGTFPOEJWEGG
|
9.3 | Kd | 149 | — | |
MLDQJTXFUGDVEO
|
8.5 | Kd | 85 | Yes | |
RKDBIDWPRDZSFA
|
8.5 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
8.4 | Kd | 153 | — | |
DKSNLQYRZJKYOC
|
8.4 | Ki | 51 | — | |
XJSFDMGICAWQFS
|
8.4 | Ki | 60 | — | |
QONPPIZSNSSCSK
|
8.3 | Ki | 45 | Yes | |
FAYAUAZLLLJJGH
|
8.2 | Ki | 36 | Yes | |
UQJQNZHGEVLHST
|
8.1 | Ki | 15 | — | |
CFIBXVQLBVNOHW
|
8.0 | Ki | 64 | — | |
NWAUBAGBGOPJLF
|
8.0 | Ki | 51 | Yes | |
WFTZMAAMCVPJJT
|
8.0 | Ki | 26 | — | |
XKZINYYXWJEYEL
|
8.0 | Ki | 37 | — | |
XOOAAYRIVATZNM
|
8.0 | Ki | 55 | — | |
IKENQUDOTQBCJH
|
8.0 | Kd | 18 | — | |
BHSOPYVVEZFHDB
|
7.9 | Ki | 25 | Yes | |
GSXRCPJTNIGKSZ
|
7.9 | Ki | 43 | — | |
KYACBMRLQMEIAI
|
7.9 | Ki | 30 | — | |
MCCCQFAOMZMZKE
|
7.9 | Ki | 52 | — | |
PTVPBWWDGZSEAF
|
7.9 | Ki | 63 | — | |
ULHGAQSVFPOUDY
|
7.9 | Ki | 43 | — | |
UOOZSMNSBYVUGZ
|
7.9 | Ki | 32 | — | |
ZXLFIHLBHMLHFJ
|
7.9 | Ki | 31 | — | |
AGYRJOAGMDIFKL
|
7.8 | Ki | 17 | — | |
PUPCRRRSBUYJAD
|
7.8 | Ki | 44 | Yes | |
SFPWNTQWFFNJIH
|
7.8 | Ki | 48 | — | |
GCBJDOWIQHMCMR
|
7.7 | Ki | 84 | — | |
LGHBDVLAHHANMX
|
7.7 | Ki | 53 | — | |
NRGYZNJPCGRCLV
|
7.7 | Ki | 52 | — | |
WPHKIQPVPYJNAX
|
7.7 | Ki | 81 | — | |
RBXYGQNZRVPDNB
|
7.6 | Ki | 34 | — | |
UMTWTCVTRDYHQQ
|
7.6 | Ki | 56 | — | |
LCGSWTFWYNYUKS
|
7.5 | Ki | 26 | — | |
MQRDVGBWWVWMEN
|
7.5 | Ki | 47 | — | |
RQJIDUOCLNMUHR
|
7.5 | Ki | 15 | — | |
VKBFHTIUXUCYRQ
|
7.5 | Ki | 66 | — | |
ACNCCUVYXQGPKZ
|
7.4 | Ki | 31 | — | |
RWEHAHIEUDLKGT
|
7.4 | Ki | 33 | — | |
SEVCBWKJSOLMNQ
|
7.4 | Ki | 38 | — | |
XYXLUJQBBIBJFV
|
7.4 | Ki | 36 | — | |
MPVGZUGXCQEXTM
|
7.3 | Kd | 61 | Yes | |
MFMXAWQGPQXDRJ
|
7.3 | Ki | 27 | — | |
NEWAULHLLUCDPD
|
7.3 | Ki | 27 | — | |
VQPBIJGXSXEOCU
|
7.3 | Ki | 24 | — | |
BSFNGHCTZDCQBF
|
7.2 | Ki | 93 | — | |
DZSUJUOJJJCWGG
|
7.2 | Ki | 55 | Yes | |
JCZBWICLNFNCMR
|
7.2 | Ki | 9 | — | |
LXVBELDBJGYFEM
|
7.2 | Ki | 20 | — | |
YMIJUBCSOKSFRU
|
7.2 | Ki | 87 | — | |
GWMATETWMAQOFL
|
7.1 | Ki | 36 | — |