Target Details
| UniProt AC | Q8NBP7 |
|---|---|
| Gene Symbol | PCSK9 |
| Protein Name | Proprotein convertase subtilisin/kexin type 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05922 (Inhibitor_I9) PF18459 (PCSK9_C1) PF18464 (PCSK9_C2) PF18463 (PCSK9_C3) PF00082 (Peptidase_S8) |
Summary
- Multi-target molecules 227
- Clinical molecules 0
- Avg pChEMBL 6.86
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (227)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDEQYXISVCQQMO
|
6.3 | IC50 | 2 | — | |
RXGJEHGKLXXJLS
|
6.3 | IC50 | 2 | — | |
SNBPWJVDOPZESG
|
6.3 | IC50 | 2 | — | |
TYAQBURXLGATKD
|
6.3 | IC50 | 2 | — | |
TYIYZRBWVAEQDY
|
6.3 | IC50 | 2 | — | |
ULJDGEPOAMADRJ
|
6.3 | IC50 | 2 | — | |
VGPQXXHISQYBNH
|
6.3 | IC50 | 2 | — | |
VNNSUPKAKVZRAS
|
6.3 | IC50 | 2 | — | |
WKJXNKGPJMUFPV
|
6.3 | IC50 | 2 | — | |
WVBBQINPROFUTD
|
6.3 | IC50 | 2 | — | |
XDEISTVXIHIEEY
|
6.3 | IC50 | 2 | — | |
XLZSMKCEQYOUBB
|
6.3 | IC50 | 2 | — | |
XSFJGBZVNFHACL
|
6.3 | IC50 | 2 | — | |
XSICDJDMSHRDIV
|
6.3 | IC50 | 2 | — | |
XXFKDDJGZGVTLW
|
6.3 | IC50 | 2 | — | |
XZABVPJOOVOYTI
|
6.3 | IC50 | 2 | — | |
ZFWIQMUIHYZSOF
|
6.3 | IC50 | 2 | — | |
VOAMXMMBZJDXSU
|
6.2 | Ki | 2 | — | |
NHJUFNWIIVOTIH
|
6.2 | IC50 | 2 | — | |
ORPZALWAWWEEDP
|
6.2 | Kd | 2 | — | |
FPILCJQVCVIRHQ
|
6.2 | IC50 | 2 | — | |
AVCCKFHOOJRTCR
|
6.1 | IC50 | 2 | — | |
FDTXHWQFIXYHCL
|
6.1 | IC50 | 79 | — | |
TYKXIBLBQNRTJM
|
6.1 | IC50 | 2 | — | |
CZJIXNHTVSHQML
|
6.1 | IC50 | 79 | — | |
ZCBJOOXWTIJJTO
|
6.0 | IC50 | 79 | — | |
SGJYNXWRJNILLN
|
6.0 | Ki | 2 | — |